SCHEMBL7015665

SCHEMBL7015665

CCC(=O)NNC(=O)CCc1cc(N2CCOCC2)cc(NC(=O)OC(C)(C)C)n1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 11/20 0.48
NPY1R P25929 11/20 0.43
BRD4 O60885 1/20 0.38
PRKDC P78527 1/20 0.38
RAB9A P51151 1/20 0.37
AKT1 P31749 1/20 0.37
MAPT P10636 3/20 0.37
MEN1 O00255 1/20 0.36
CYP2C19 P33261 1/20 0.36
KMT2A Q03164 1/20 0.36
JAK3 P52333 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7015058 0.89 KCNH2 (0.47) KCNH2NPY1RBRD4PRKDCAKT1
SCHEMBL7018612 0.88 KCNH2 (0.49) KCNH2NPY1RBRD4PRKDCAKT1
SCHEMBL7016743 0.87 KCNH2 (0.48) KCNH2NPY1RBRD4PRKDCAKT1
SCHEMBL12946506 0.83 KCNH2 (0.48) KCNH2NPY1RBRD4PRKDCRAB9A
SCHEMBL7016153 0.83 KCNH2 (0.48) KCNH2NPY1RBRD4PRKDCRAB9A
SCHEMBL7015881 0.81 KCNH2 (0.51) KCNH2NPY1RBRD4PRKDCMAPT
SCHEMBL960822 0.79 KCNH2 (0.77) KCNH2NPY1RBRD4PRKDC
SCHEMBL7015353 0.79 KCNH2 (0.56) KCNH2NPY1RBRD4PRKDC
SCHEMBL7019934 0.78 NPY1R (0.61) KCNH2NPY1R
SCHEMBL7020498 0.77 KCNH2 (0.41) KCNH2NPY1RBRD4PRKDCRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889034-B1 AMINOPYRIDINE DERIVATIVES BANYU PHARMA CO LTD (JP) 2003-09-17 EP disclosed
US-6011039-A USEFUL AS NEUROPEPTIDE Y RECEPTOR ANTAGONISTS; TREATING HYPERPHAGIA, OBESITY OR DIABETES BANYU PHARMACEUTICAL CO., LTD. (JP) 2000-01-04 US disclosed
EP-0889034-A1 AMINOPYRIDINE DERIVATIVES BANYU PHARMACEUTICAL CO., LTD. (JP) 1999-01-07 EP disclosed