SCHEMBL7016153

SCHEMBL7016153

CC(C)(C)OC(=O)Nc1cc(N2CCOCC2)cc(CO)n1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 9/20 0.48
PRKDC P78527 1/20 0.43
BRD4 O60885 2/20 0.43
NPY1R P25929 8/20 0.42
MAPT P10636 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
KMT2A Q03164 1/20 0.39
CD274 Q9NZQ7 1/20 0.39
GAA P10253 1/20 0.38
MTOR P42345 2/20 0.38
PIK3CA P42336 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
EGFR P00533 1/20 0.38
AKT1 P31749 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12946506 0.91 KCNH2 (0.48) KCNH2PRKDCBRD4NPY1RMAPT
SCHEMBL7018612 0.87 KCNH2 (0.49) KCNH2PRKDCBRD4NPY1RMAPT
SCHEMBL503981 0.87 KCNQ3 (0.36) KCNH2BRD4NPY1RKDM4E
SCHEMBL7016743 0.86 KCNH2 (0.48) KCNH2PRKDCBRD4NPY1RMAPT
SCHEMBL7015058 0.85 KCNH2 (0.47) KCNH2PRKDCBRD4NPY1RMAPT
SCHEMBL7015665 0.83 KCNH2 (0.48) KCNH2PRKDCBRD4NPY1RMAPT
SCHEMBL113716 0.82 KCNH2 (0.41) KCNH2PRKDCBRD4NPY1RMAPT
SCHEMBL7015881 0.82 KCNH2 (0.51) KCNH2PRKDCBRD4NPY1RMAPT
SCHEMBL7020498 0.82 KCNH2 (0.41) KCNH2PRKDCBRD4NPY1RMAPT
SCHEMBL962372 0.82 PRKDC (0.43) KCNH2PRKDCBRD4MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889034-B1 AMINOPYRIDINE DERIVATIVES BANYU PHARMA CO LTD (JP) 2003-09-17 EP disclosed
US-6011039-A USEFUL AS NEUROPEPTIDE Y RECEPTOR ANTAGONISTS; TREATING HYPERPHAGIA, OBESITY OR DIABETES BANYU PHARMACEUTICAL CO., LTD. (JP) 2000-01-04 US disclosed
EP-0889034-A1 AMINOPYRIDINE DERIVATIVES BANYU PHARMACEUTICAL CO., LTD. (JP) 1999-01-07 EP disclosed