SCHEMBL7016018

SCHEMBL7016018

Cc1nc2c(O)cccn2c(=O)c1C

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.56
KDM4E B2RXH2 6/20 0.56
GAA P10253 5/20 0.56
LMNA P02545 1/20 0.56
GLA P06280 1/20 0.56
MPI P34949 1/20 0.56
ADRA2A P08913 1/20 0.43
ADRA2B P18089 1/20 0.43
ADRA2C P18825 1/20 0.43
ADRA1A P35348 1/20 0.43
HTR1A P08908 1/20 0.43
DRD2 P14416 1/20 0.43
HTR2A P28223 1/20 0.43
CASR P41180 1/20 0.41
HPGD P15428 4/20 0.40
MAPT P10636 3/20 0.40
MEN1 O00255 1/20 0.40
POLB P06746 1/20 0.40
BLM P54132 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11807279 0.83 KDM4E (0.55) ALDH1A1KDM4EGAALMNAHPGD
SCHEMBL2902371 0.81 KDM4E (0.51) ALDH1A1KDM4EGAALMNAGLA
SCHEMBL15519297 0.81 KDM4E (0.40) ALDH1A1KDM4EGAALMNAGLA
Hydrochloric Acid SCHEMBL11357932 0.80 KDM4E (0.54) ALDH1A1KDM4EGAALMNAGLA
SCHEMBL7886328 0.79 ADRA2A (0.53) ALDH1A1KDM4EGAALMNAGLA
SCHEMBL900644 0.79 ADRA2A (0.53) ALDH1A1KDM4EGAALMNAGLA
SCHEMBL900661 0.79 ADRA2A (0.55) ALDH1A1KDM4EGAALMNAGLA
SCHEMBL4063787 0.79 ALDH1A1 (0.54) ALDH1A1KDM4EGAALMNAGLA
SCHEMBL2899691 0.78 MAPT (0.55) ALDH1A1KDM4EGAALMNAGLA
Hydrochloric Acid SCHEMBL900773 0.78 ADRA2A (0.52) ALDH1A1KDM4EGAALMNAGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed