SCHEMBL7016076

SCHEMBL7016076

CCc1cccc2nc(SCc3ccc(C(=O)c4ccc([N+](=O)[O-])cc4)cc3)n(C)c(=O)c12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.49
MEN1 O00255 5/20 0.49
KMT2A Q03164 5/20 0.49
RAB9A P51151 2/20 0.49
NPC1 O15118 1/20 0.49
LMNA P02545 4/20 0.49
L3MBTL1 Q9Y468 2/20 0.49
USP2 O75604 1/20 0.49
MAPT P10636 5/20 0.48
SMN1; SMN2 Q16637 5/20 0.48
POLB P06746 2/20 0.48
NPSR1 Q6W5P4 2/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
TP53 P04637 1/20 0.45
KDM4E B2RXH2 1/20 0.45
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7017243 0.90 MAPT (0.50) ALDH1A1MEN1KMT2ARAB9ANPC1
SCHEMBL7014213 0.87 DRD2 (0.48) ALDH1A1MEN1KMT2ALMNAMAPT
SCHEMBL7017967 0.85 DAO (0.52) ALDH1A1MEN1KMT2ARAB9ANPC1
SCHEMBL8649589 0.83 MEN1 (0.43) ALDH1A1MEN1KMT2ARAB9AL3MBTL1
SCHEMBL7011506 0.80 MEN1 (0.55) ALDH1A1MEN1KMT2AUSP2MAPT
SCHEMBL7014355 0.78 DRD2 (0.50) ALDH1A1MEN1KMT2ARAB9AMAPT
SCHEMBL7014710 0.78 TP53 (0.47) MEN1KMT2ALMNAL3MBTL1MAPT
SCHEMBL7017586 0.77 MEN1 (0.57) ALDH1A1MEN1KMT2AUSP2SMN1; SMN2
SCHEMBL7101327 0.77 MEN1 (0.60) ALDH1A1MEN1KMT2ALMNAMAPT
SCHEMBL7015787 0.77 MEN1 (0.51) ALDH1A1MEN1KMT2ANPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed