SCHEMBL7014355

SCHEMBL7014355

COCc1cccc2nc(SCc3ccc(C(=O)c4ccc(Cl)cc4)cc3)n(C)c(=O)c12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 6/20 0.50
TBXA2R P21731 6/20 0.50
MAPT P10636 2/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
HDAC9 Q9UKV0 1/20 0.44
HDAC5 Q9UQL6 1/20 0.44
PTGDR2 Q9Y5Y4 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7014710 0.91 TP53 (0.47) MAPTCYP2C9CYP2C19MEN1KMT2A
SCHEMBL7014213 0.91 DRD2 (0.48) DRD2TBXA2RMAPTCYP1A2CYP2D6
SCHEMBL7012515 0.88 NLRP3 (0.43) DRD2TBXA2RMAPTHDAC3HDAC4
SCHEMBL7014904 0.88 LMNA (0.45) DRD2TBXA2RMAPTCYP1A2CYP2D6
SCHEMBL7018370 0.85 MEN1 (0.50) DRD2TBXA2RMAPTCYP1A2CYP2D6
SCHEMBL7010850 0.85 DRD2 (0.55) DRD2TBXA2RMAPTCYP1A2CYP2D6
SCHEMBL7017967 0.83 DAO (0.52) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL8649589 0.81 MEN1 (0.43) DRD2TBXA2RMAPTHDAC3HDAC4
SCHEMBL7015339 0.80 KMT2A (0.68) DRD2TBXA2RMAPTCYP1A2CYP2D6
SCHEMBL7011506 0.80 MEN1 (0.55) MAPTCYP1A2CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed