SCHEMBL7016170

SCHEMBL7016170

O=c1nc[nH]c2occc12

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 12/20 0.33
PIM1 P11309 4/20 0.33
PDPK1 O15530 2/20 0.33
PIM3 Q86V86 2/20 0.33
CHEK1 O14757 2/20 0.33
AKT1 P31749 1/20 0.33
FLT3 P36888 1/20 0.33
CA12 O43570 1/20 0.33
ALOX15 P16050 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CA9 Q16790 1/20 0.33
TNKS2 Q9H2K2 1/20 0.33
CDC7 O00311 1/20 0.31
CSNK2A2 P19784 1/20 0.31
CSNK2B P67870 1/20 0.31
CSNK2A1 P68400 1/20 0.31
CSNK2A3 Q8NEV1 1/20 0.31
PIM2 Q9P1W9 1/20 0.31
KDM4E B2RXH2 1/20 0.31
KDM4A O75164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2976500 0.68 PARP1 (0.46) PARP1PIM1PDPK1PIM3CHEK1
SCHEMBL1550252 0.68 KDM4E (0.31) KDM4EALDH1A1AURKA
SCHEMBL4240700 0.67 CCR8 (0.46) SMN1; SMN2KDM4ENFKB1MAOAMAOB
SCHEMBL15707647 0.63 GSK3B (0.41) PARP1PIM1PDPK1PIM3CHEK1
Quinazolinone SCHEMBL10418 0.63 PARP1 (0.48) PARP1PIM1PDPK1CHEK1CA12
SCHEMBL19153215 0.62 MAOA (0.42) PARP1PIM1PDPK1PIM3CHEK1
Quinazolinone SCHEMBL7746268 0.61 PARP1 (0.47) PARP1PIM1PDPK1CHEK1CA12
Quinazolinone SCHEMBL8201415 0.61 PARP1 (0.47) PARP1PIM1PDPK1CHEK1CA12
SCHEMBL7015716 0.61 PNP (0.32) PARP1PIM1PDPK1PIM3CHEK1
SCHEMBL19743069 0.60 PARP1 (0.40) PARP1PIM1SMN1; SMN2CSNK2A2CSNK2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP claimed
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed