SCHEMBL7016244

SCHEMBL7016244

C=Cc1ccc(S(=O)(=O)C2(N(C)C(=O)CC)CCN(c3ccncc3)CC2)cc1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.41
CYP2D6 P10635 3/20 0.41
CYP2C19 P33261 3/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2C9 P11712 4/20 0.38
CYP3A4 P08684 4/20 0.38
HIF1A Q16665 3/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
F10 P00742 4/20 0.37
MMP2 P08253 3/20 0.36
MMP13 P45452 3/20 0.36
ITGB3 P05106 4/20 0.35
ITGA2B P08514 4/20 0.35
ADAM17 P78536 1/20 0.35
CYP17A1 P05093 1/20 0.35
CYP21A2 P08686 1/20 0.35
CYP19A1 P11511 1/20 0.35
CYP11B1 P15538 1/20 0.35
RORC P51449 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7013734 0.80 F10 (0.57) F10
SCHEMBL7017519 0.70 F10 (0.47) F10
Hydrochloric Acid SCHEMBL7017062 0.69 F10 (0.57) F10
SCHEMBL6888024 0.67 MEN1 (0.45) TSHRCYP2D6CYP2C19CYP1A2CYP2C9
Hydrochloric Acid SCHEMBL6896243 0.66 MEN1 (0.45) TSHRCYP2D6CYP2C19CYP1A2CYP2C9
SCHEMBL6751594 0.62 TDP1 (0.78) TSHRCYP2D6SMN1; SMN2
SCHEMBL24378028 0.61 CYP17A1 (0.57) TSHRCYP2D6CYP2C19CYP1A2CYP2C9
Propionic Acid SCHEMBL28801703 0.61 JUN (0.40) CYP2C19CYP1A2SMN1; SMN2
SCHEMBL3315322 0.61 CYP2C9 (0.51) TSHRCYP2D6CYP2C19CYP1A2CYP2C9
SCHEMBL30593971 0.60 CHKA (0.55) TSHRCYP2D6CYP2C19CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030187023-A1 Sulfone derivatives, process for their production and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2003-10-02 US disclosed
EP-1302462-A1 SULFONE DERIVATIVES, PROCESS FOR THEIR PRODUCTION AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2003-04-16 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030187023-A1 Sulfone derivatives, process for their production and use thereof SULT1E1, RRS1, SHH TSHR 1149/4885CYP2D6 332/4885CYP2C19 1061/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.