SCHEMBL7016460

SCHEMBL7016460

COc1ccc(C(=O)O)c(C(N)=O)c1

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.57
ALDH1A1 P00352 3/20 0.53
AKR1C3 P42330 9/20 0.53
AKR1C2 P52895 9/20 0.53
KDM4E B2RXH2 5/20 0.53
POLB P06746 2/20 0.53
PARP1 P09874 2/20 0.50
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
GAA P10253 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
PARP10 Q53GL7 1/20 0.50
PARP2 Q9UGN5 1/20 0.50
PARP4 Q9UKK3 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2835948 0.90 PARP1 (0.55) SMN1; SMN2ALDH1A1KDM4EPARP1NPC1
SCHEMBL383820 0.88 ALDH1A1 (0.66) SMN1; SMN2ALDH1A1AKR1C3AKR1C2KDM4E
Benzene SCHEMBL29227606 0.86 ALDH1A1 (0.63) SMN1; SMN2ALDH1A1AKR1C3AKR1C2KDM4E
SCHEMBL26768695 0.86 SMN1; SMN2 (0.68) SMN1; SMN2ALDH1A1AKR1C3AKR1C2KDM4E
SCHEMBL30629168 0.86 SMN1; SMN2 (0.68) SMN1; SMN2ALDH1A1AKR1C3AKR1C2KDM4E
SCHEMBL3277227 0.85 ALDH1A1 (0.62) SMN1; SMN2ALDH1A1KDM4EPARP1NPC1
SCHEMBL3037245 0.83 ALDH1A1 (0.65) SMN1; SMN2ALDH1A1AKR1C3AKR1C2KDM4E
SCHEMBL15317994 0.81 POLB (0.58) ALDH1A1KDM4EPOLBTDP1L3MBTL1
SCHEMBL11780068 0.81 POLB (0.58) ALDH1A1KDM4EPOLBTDP1L3MBTL1
SCHEMBL1956889 0.81 KDM4E (0.60) SMN1; SMN2ALDH1A1AKR1C3AKR1C2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1370562-A1 THIENO[2,3-D]PYRIMIDINDIONE DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS Warner-Lambert Company LLC (US) 2003-12-17 EP disclosed
WO-2002064598-A1 THIENO'2,3-D PYRIMIDINDIONE DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2002-08-22 WO disclosed