SCHEMBL7016797

SCHEMBL7016797

COc1ccc2ccc(OC)c(CCNC(C)=O)c2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 15/20 0.77
MTNR1B P49286 14/20 0.77
HTR2C P28335 1/20 0.65
HTR2B P41595 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18317861 0.91 MTNR1A (0.67) MTNR1AMTNR1BHTR2CHTR2B
SCHEMBL7014618 0.90 MTNR1A (0.64) MTNR1AMTNR1B
SCHEMBL7022938 0.87 MTNR1A (0.59) MTNR1AMTNR1B
SCHEMBL7336150 0.86 MTNR1A (0.64) MTNR1AMTNR1BHTR2CHTR2B
SCHEMBL29032224 0.86 MTNR1A (0.64) MTNR1AMTNR1BHTR2CHTR2B
SCHEMBL18317974 0.84 MTNR1A (0.60) MTNR1AMTNR1BHTR2CHTR2B
SCHEMBL8186004 0.84 MTNR1A (0.61) MTNR1AMTNR1BHTR2CHTR2B
SCHEMBL19638479 0.83 MTNR1A (0.63) MTNR1AMTNR1BHTR2CHTR2B
SCHEMBL18318761 0.83 MTNR1A (0.55) MTNR1AMTNR1BHTR2CHTR2B
SCHEMBL9119468 0.80 MTNR1A (0.67) MTNR1AMTNR1BHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1181050-C Novel substituted dimeric compounds, its preparing process and medicinal compsns. containing same ɪά��ʵ���� 2004-12-22 CN disclosed
US-6635650-B2 Such as N-(2-(7-(2-((8-(2-(acetyl-amino)ethyl)-2-naphthyl) oxy)ethoxy)-1-napthyl)ethyl)acetamide for treating or preventing melatoninergic disorders LES LABORATOIRES SERVIER (FR) 2003-10-21 US disclosed
EP-1038863-B1 Substituted dimeric compounds, process for their preparation and pharmaceutical compositions thereof SERVIER LAB (FR) 2003-06-04 EP disclosed
US-20020035114-A1 Substituted dimeric compounds LESIEUR DANIEL (FR) 2002-03-21 US disclosed
US-6319930-B1 CONTAINING FUSED AROMATIC CARBO- OR HETEROCYCLIC RINGS AND AMIDE, THIOAMIDE, UREA OR THIOUREA GROUPS; USEFUL IN TREATING OR IN PREVENTING MELATONINERGIC DISORDERS. ADIR ET COMPAGNIE (FR) 2001-11-20 US disclosed
CN-1273967-A Novel substituted dimeric compounds, its preparing process and medicinal compsns. containing same ADIR (FR) 2000-11-22 CN disclosed
EP-1038863-A2 Substituted dimeric compounds, process for their preparation and pharmaceutical compositions thereof ADIR ET COMPAGNIE (FR) 2000-09-27 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020035114-A1 Substituted dimeric compounds NR0B2, NR0B1, NR2C2 MTNR1A 4/4885MTNR1B 5/4885HTR2C 191/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.