SCHEMBL7017472

SCHEMBL7017472

CC(C)(CC(N)=O)CC(=O)N(CCCC#N)C1CCNC1

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 18/20 0.37
SLC6A2 P23975 16/20 0.37
SLC6A3 Q01959 8/20 0.37
KCNH2 Q12809 3/20 0.33
DPP4 P27487 2/20 0.33
CYP2D6 P10635 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7020799 0.82 SLC6A2 (0.36) SLC6A4SLC6A2SLC6A3KCNH2
SCHEMBL7018597 0.77 SLC6A4 (0.37) SLC6A4SLC6A2SLC6A3KCNH2DPP4
SCHEMBL7425515 0.75 SLC6A2 (0.40) SLC6A4SLC6A2SLC6A3KCNH2CYP2D6
SCHEMBL7417580 0.71 DPP4 (0.30) DPP4
SCHEMBL5987555 0.69 PTGS1 (0.34) SLC6A4KCNH2DPP4
SCHEMBL28246290 0.63 SLC6A2 (0.47) SLC6A4SLC6A2SLC6A3KCNH2CYP2D6
SCHEMBL1221462 0.63 SLC6A2 (0.47) SLC6A4SLC6A2SLC6A3KCNH2CYP2D6
SCHEMBL3821799 0.63 SLC6A2 (0.47) SLC6A4SLC6A2SLC6A3KCNH2CYP2D6
SCHEMBL22878185 0.63 NOS2 (0.40) SLC6A4SLC6A2SLC6A3
SCHEMBL27957684 0.63 SLC6A2 (0.50) SLC6A4SLC6A2SLC6A3KCNH2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2003529546-A 2003-10-07 JP claimed
EP-1218372-A1 NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES Boehringer Ingelheim Pharmaceuticals, Inc. (US) 2002-07-03 EP claimed
WO-2001019816-A1 NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2001-03-22 WO claimed
EP-1218372-A1 NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES Boehringer Ingelheim Pharmaceuticals, Inc. (US) 2002-07-03 EP disclosed
WO-2001019816-A1 NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2001-03-22 WO disclosed