SCHEMBL7017658

SCHEMBL7017658

O=c1c2cc(Cl)ccc2nc2n1C[C@H](CS)S2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP1B1 Q16678 1/20 0.39
KDM4E B2RXH2 3/20 0.39
HTT P42858 3/20 0.39
LMNA P02545 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
HSD17B10 Q99714 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
MAPT P10636 2/20 0.37
MAPK1 P28482 1/20 0.37
APP P05067 1/20 0.35
TUBB4A P04350 2/20 0.35
TUBB P07437 2/20 0.35
TUBA3C P0DPH7 2/20 0.35
TUBA1B P68363 2/20 0.35
TUBA4A P68366 2/20 0.35
TUBB4B P68371 2/20 0.35
TUBB3 Q13509 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6804059 0.90 KMT2A (0.40) CYP1A1CYP1A2CYP1B1KDM4EHTT
SCHEMBL6804062 0.90 KMT2A (0.40) CYP1A1CYP1A2CYP1B1KDM4EHTT
SCHEMBL6700295 0.90 KMT2A (0.40) CYP1A1CYP1A2CYP1B1KDM4EHTT
SCHEMBL6701095 0.82 ALDH1A1 (0.49) CYP1A2KDM4EHTTLMNAL3MBTL1
SCHEMBL6804691 0.82 ALDH1A1 (0.49) CYP1A2KDM4EHTTLMNAL3MBTL1
SCHEMBL6702099 0.78 CYP1A1 (0.39) CYP1A1CYP1A2CYP1B1KDM4EHTT
SCHEMBL7000926 0.78 CYP1A1 (0.39) CYP1A1CYP1A2CYP1B1KDM4EHTT
SCHEMBL7015998 0.73 PDE7A (0.40) HTTL3MBTL1SMN1; SMN2ALDH1A1
SCHEMBL7019520 0.72 RAB9A (0.53) CYP1A2KDM4EHTTLMNAHSD17B10
SCHEMBL7018731 0.70 MAPT (0.51) CYP1A2KDM4EHTTLMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003089416-A1 SUBSTITUTED PYRIMIDINE-2,4(1H,3H)-DIONES FOR USE AS MATRIX METALLOPROTEINASE (MMP) INHIBITORS IBFB GMBH (DE) 2003-10-30 WO disclosed
EP-1357114-A1 Substituted pyrimidin-2,4(1H,3H)-diones as inhibitors of Matrix Metalloproteinases (MMP) IBFB GmbH Privates Institut für biomedizinische Forschung und Beratung (DE) 2003-10-29 EP disclosed