SCHEMBL7017706

SCHEMBL7017706

Cn1c(S)nc2ncn(C)c2c1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 5/20 0.47
ADORA2A P29274 3/20 0.47
GDA Q9Y2T3 2/20 0.47
PIK3CD O00329 1/20 0.47
POLB P06746 1/20 0.47
ADORA3 P0DMS8 1/20 0.47
CNR1 P21554 1/20 0.47
ACHE P22303 1/20 0.47
ADORA1 P30542 1/20 0.47
NTSR1 P30989 1/20 0.47
MC3R P41968 1/20 0.47
NOTUM Q6P988 1/20 0.47
SIRT3 Q9NTG7 1/20 0.47
NR2E1 Q9Y466 1/20 0.47
CYP3A4 P08684 3/20 0.45
PMP22 Q01453 3/20 0.45
BLM P54132 2/20 0.45
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45
MAPT P10636 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21393459 0.80 ADORA2B (0.49) ADORA2BADORA2AGDAPIK3CDPOLB
SCHEMBL21961 0.79 ADORA2B (0.47) ADORA2BADORA2AGDAPIK3CDPOLB
SCHEMBL31288035 0.79 ADORA2B (0.47) ADORA2BADORA2AGDAPIK3CDPOLB
Hydrochloric Acid SCHEMBL17186276 0.77 ADORA2A (0.46) ADORA2BADORA2AGDAPIK3CDPOLB
SCHEMBL31646363 0.76 ADORA2B (0.45) ADORA2BADORA2AGDAPIK3CDPOLB
SCHEMBL20203174 0.74 ADORA2A (0.48) ADORA2BADORA2AGDAPIK3CDPOLB
SCHEMBL9466617 0.72 ADORA2A (0.38) ADORA2BADORA2AGDAPIK3CDPOLB
SCHEMBL21363449 0.69 ADORA2A (0.38) ADORA2BADORA2AGDAPIK3CDPOLB
SCHEMBL2775208 0.68 GDA (0.32) ADORA2BADORA2AGDAPIK3CDPOLB
SCHEMBL21367881 0.68 ADORA2B (0.40) ADORA2BADORA2AGDAPIK3CDPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed