SCHEMBL7019135

SCHEMBL7019135

CCOC(=O)C1=C(C)N=CCC1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.39
CYP1A2 P05177 2/20 0.39
GAA P10253 2/20 0.38
TSHR P16473 1/20 0.38
ALDH1A1 P00352 3/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
LMNA P02545 2/20 0.36
CASP1 P29466 1/20 0.36
CA12 O43570 3/20 0.36
CA1 P00915 3/20 0.36
CA2 P00918 3/20 0.36
CA7 P43166 3/20 0.36
CA9 Q16790 3/20 0.36
CA14 Q9ULX7 3/20 0.36
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6885396 0.85 MAPT (0.38) MAPTCYP1A2GAATSHRALDH1A1
SCHEMBL10707078 0.70 SMN1; SMN2 (0.39) MAPTCYP1A2GAATSHRALDH1A1
SCHEMBL4773450 0.70 CYP1A2 (0.39) MAPTCYP1A2GAATSHRALDH1A1
SCHEMBL22249801 0.69 MAPT (0.38) MAPTCYP1A2GAATSHRALDH1A1
SCHEMBL6616099 0.68 MAPT (0.40) MAPTCYP1A2GAATSHRALDH1A1
SCHEMBL9626490 0.67 ALDH1A1 (0.49) MAPTCYP1A2GAATSHRALDH1A1
SCHEMBL17842993 0.67 CYP1A2 (0.39) MAPTCYP1A2GAATSHRALDH1A1
SCHEMBL10243639 0.66 ALDH1A1 (0.38) MAPTCYP1A2GAATSHRALDH1A1
SCHEMBL5057759 0.64 MEN1 (0.42) MAPTCYP1A2GAATSHRALDH1A1
SCHEMBL29150933 0.64

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2726479-A1 NOVEL INHIBITOR COMPOUNDS OF PHOSPHODIESTERASE TYPE 10A AbbVie Deutschland GmbH & Co KG (DE) 2014-05-07 EP disclosed
WO-2013000994-A1 NOVEL INHIBITOR COMPOUNDS OF PHOSPHODIESTERASE TYPE 10A ABBOTT GMBH & CO. KG (DE) 2013-01-03 WO disclosed
EP-1309565-A1 HETEROCYCLIC MUTILIN ESTERS AND THEIR USE AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2003-05-14 EP disclosed
WO-2002012199-A1 HETEROCYCLIC MUTILIN ESTERS AND THEIR USE AS ANTIBACTERIALS SMITHKLINE BEECHAM P.L.C. (GB) 2002-02-14 WO disclosed