SCHEMBL7019303

SCHEMBL7019303

CSc1nc2c(ccn2Cc2ccc(C(=O)c3ccc(Cl)cc3)cc2)c(=O)n1CCO

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.46
TDP1 Q9NUW8 1/20 0.46
ATM Q13315 1/20 0.44
APOBEC3G Q9HC16 1/20 0.44
KMT2A Q03164 2/20 0.43
RXFP1 Q9HBX9 2/20 0.41
HDAC1 Q13547 4/20 0.40
HDAC6 Q9UBN7 4/20 0.40
HDAC4 P56524 2/20 0.40
MAPT P10636 4/20 0.39
HDAC2 Q92769 3/20 0.39
HDAC3 O15379 2/20 0.39
HDAC8 Q9BY41 2/20 0.39
FYN P06241 1/20 0.39
SRC P12931 1/20 0.39
FLT3 P36888 1/20 0.39
TSHR P16473 2/20 0.37
ALDH1A1 P00352 2/20 0.37
MAPK1 P28482 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7014404 0.92 TP53 (0.46) TP53TDP1ATMAPOBEC3GKMT2A
SCHEMBL7017888 0.90 TP53 (0.47) TP53TDP1ATMAPOBEC3GKMT2A
SCHEMBL7018715 0.89 TP53 (0.48) TP53TDP1ATMAPOBEC3GKMT2A
SCHEMBL7008875 0.88 TP53 (0.42) TP53TDP1ATMAPOBEC3GKMT2A
SCHEMBL7019301 0.83 TP53 (0.45) TP53TDP1ATMAPOBEC3GKMT2A
SCHEMBL7019933 0.82 HDAC1 (0.41) TP53TDP1KMT2ARXFP1HDAC1
SCHEMBL7008873 0.79 TP53 (0.42) TP53TDP1ATMAPOBEC3GKMT2A
SCHEMBL7010809 0.76 TP53 (0.48) TP53TDP1ATMAPOBEC3GKMT2A
SCHEMBL7015809 0.76 HDAC6 (0.48) TP53KMT2AHDAC1HDAC6HDAC4
SCHEMBL7018264 0.76 BCL6 (0.48) TP53TDP1KMT2ARXFP1HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed