SCHEMBL7019374

SCHEMBL7019374

NC(=O)c1ccc(Cc2ncc[nH]2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 4/20 0.57
CYP17A1 P05093 1/20 0.51
PLA2G10 O15496 1/20 0.50
PLA2G2A P14555 1/20 0.50
PARP10 Q53GL7 2/20 0.44
KLK1 P06870 1/20 0.43
KLK5 Q9Y337 1/20 0.43
HTR1A P08908 1/20 0.43
GAA P10253 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
IKBKB O14920 1/20 0.41
CHUK O15111 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
TBXAS1 P24557 2/20 0.40
HDAC3 O15379 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
NCOR2 Q9Y618 1/20 0.39
MKNK1 Q9BUB5 1/20 0.39
MKNK2 Q9HBH9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11357644 0.87 TAAR1 (0.61) TAAR1HTR1AGAASMN1; SMN2NPC1
SCHEMBL7022457 0.86 TBXAS1 (0.45) TAAR1CYP17A1PLA2G10PLA2G2APARP10
Hydrochloric Acid SCHEMBL9853948 0.84 TAAR1 (0.62) TAAR1KLK1KLK5HTR1AGAA
SCHEMBL6432418 0.84 TAAR1 (0.57) TAAR1KLK1KLK5HTR1AGAA
SCHEMBL13372830 0.82 TAAR1 (0.80) TAAR1HTR1ASMN1; SMN2
SCHEMBL6746541 0.80 ALDH1A1 (0.60) TAAR1HTR1AGAASMN1; SMN2NPC1
SCHEMBL10944433 0.79 PARP1 (0.54) TAAR1PLA2G10PLA2G2APARP10HTR1A
SCHEMBL10999093 0.79 TAAR1 (0.55) TAAR1HTR1AGAASMN1; SMN2RAB9A
SCHEMBL10945831 0.79 TAAR1 (0.51) TAAR1HTR1AGAASMN1; SMN2RAB9A
SCHEMBL9416067 0.79 TAAR1 (0.64) TAAR1HTR1AGAASMN1; SMN2TBXAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1325006-A2 HETEROCYCLIC COMPOUNDS AS LIGANDS OF THE GABA A? RECEPTOR NEUROGEN CORPORATION (US) 2003-07-09 EP claimed
WO-2002012442-A2 HETEROCYCLIC COMPOUNDS AS LIGANDS OF THE GABAA RECEPTOR NEUROGEN CORPORATION (US) 2002-02-14 WO claimed