SCHEMBL7019465

SCHEMBL7019465

SC(=NCCc1ccccc1)Nc1ccc(Oc2ccc(NC(S)=NCCc3ccccc3)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 4/20 0.49
HDAC1 Q13547 2/20 0.47
KMT2A Q03164 4/20 0.47
MEN1 O00255 3/20 0.47
GAA P10253 2/20 0.47
POLB P06746 1/20 0.47
RECQL P46063 1/20 0.45
RNF4 P78317 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
LMNA P02545 1/20 0.43
TP53 P04637 1/20 0.43
HPGD P15428 2/20 0.42
PGR P06401 1/20 0.42
ALDH1A1 P00352 2/20 0.42
NPC1 O15118 1/20 0.41
CRHBP P24387 1/20 0.41
RAB9A P51151 1/20 0.41
CRHR2 Q13324 1/20 0.41
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7025481 0.83 NPY5R (0.39) NPY5RHDAC1KMT2AMEN1GAA
SCHEMBL7896868 0.80 NPY5R (0.50) NPY5RHDAC1KMT2AMEN1GAA
SCHEMBL7898569 0.77 NPY5R (0.47) NPY5RHDAC1KMT2AMEN1GAA
SCHEMBL7895718 0.73 HPGD (0.47) HDAC1KMT2AMEN1GAAPOLB
SCHEMBL7019453 0.69 RAB9A (0.77) KMT2AMEN1GAAPOLBSMN1; SMN2
SCHEMBL10789758 0.68 CXCR4 (0.44) HDAC1GAASMN1; SMN2LMNATP53
SCHEMBL10789750 0.68 CXCR4 (0.44) HDAC1GAASMN1; SMN2LMNATP53
SCHEMBL21316586 0.67 HPGD (0.66) HDAC1RECQLRNF4SMN1; SMN2LMNA
SCHEMBL23573012 0.67 FFAR1 (0.61) FFAR1FFAR4
SCHEMBL12167954 0.67 RAB9A (0.77) HDAC1KMT2AMEN1GAARECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973735-B1 POLYAROMATIC ANTIVIRAL COMPOSITIONS UPJOHN CO (US) 2003-01-29 EP claimed
US-5958983-A NOVEL COMPOUNDS HAVING ANTIVIRAL ACTIVITY AGAINST HERPES, TOPICAL ADMINISTRATION THEM TO TREAT PATIENTS WITH HERPES; WORK BY INHIBITING THE INITIATION OF HERPES VIRAL DNA SYNTHESIS IN HOST CELLS PHARMACIA & UPJOHN COMPANY (US) 1999-09-28 US claimed
EP-0973735-B1 POLYAROMATIC ANTIVIRAL COMPOSITIONS UPJOHN CO (US) 2003-01-29 EP disclosed
EP-1148048-A2 Polyaromatic antiviral compositions PHARMACIA & UPJOHN COMPANY (US) 2001-10-24 EP disclosed
US-6147116-A TOPICALLY ADMINISTERING BENZENE DERIVATIVE SUBSTITUTED WITH UREIDO-, THIOUREIDO, AND/OR SULFONAMIDO GROUPS TO TREAT HERPES PHARMACIA & UPJOHN COMPANY (US) 2000-11-14 US disclosed
US-5958983-A NOVEL COMPOUNDS HAVING ANTIVIRAL ACTIVITY AGAINST HERPES, TOPICAL ADMINISTRATION THEM TO TREAT PATIENTS WITH HERPES; WORK BY INHIBITING THE INITIATION OF HERPES VIRAL DNA SYNTHESIS IN HOST CELLS PHARMACIA & UPJOHN COMPANY (US) 1999-09-28 US disclosed