SCHEMBL7019473

SCHEMBL7019473

NCc1ccc(O)c(C2CCN(C(=O)c3cncc(CCc4ccccc4)c3)CC2)c1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TPSAB1 Q15661 5/20 0.41
KCNH2 Q12809 4/20 0.41
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
TRPC6 Q9Y210 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
ALOX15 P16050 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
EGLN1 Q9GZT9 1/20 0.38
NUDT1 P36639 1/20 0.38
BACE1 P56817 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4404743 0.99 TPSAB1 (0.40) TPSAB1KCNH2CYP2C9CYP2C19MEN1
SCHEMBL1380988 0.90 TRPC6 (0.41) TPSAB1KCNH2CYP2C9CYP2C19MEN1
SCHEMBL1381851 0.90 TPSAB1 (0.51) TPSAB1KCNH2CYP2C9CYP2C19MEN1
Hydrochloric Acid SCHEMBL4401941 0.89 TRPC6 (0.41) TPSAB1KCNH2CYP2C9CYP2C19MEN1
Hydrochloric Acid SCHEMBL4403389 0.89 TPSAB1 (0.50) TPSAB1KCNH2CYP2C9CYP2C19MEN1
Hydrochloric Acid SCHEMBL6486065 0.89 TPSAB1 (0.50) TPSAB1KCNH2CYP2C9CYP2C19MEN1
SCHEMBL7021172 0.85 TPSAB1 (0.53) TPSAB1
Hydrochloric Acid SCHEMBL6321910 0.84 MEN1 (0.41) KCNH2CYP2C9MEN1KMT2ATRPC6
Hydrochloric Acid SCHEMBL4402047 0.84 TPSAB1 (0.52) TPSAB1
Hydrochloric Acid SCHEMBL27528148 0.84 NAMPT (0.41) TPSAB1KCNH2CYP2C9CYP2C19MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1296972-A1 ARYLMETHYLAMINE DERIVATIVES FOR USE AS TRYPTASE INHIBITORS Aventis Pharmaceuticals Inc. (US) 2003-04-02 EP disclosed
WO-2001090101-A1 ARYLMETHYLAMINE DERIVATIVES FOR USE AS TRYPTASE INHIBITORS AVENTIS PHARMACEUTICALS INC. (US) 2001-11-29 WO disclosed