SCHEMBL7019649

SCHEMBL7019649

CC(=O)OCC(C)(C)c1ccc([N+](=O)[O-])cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.52
POLB P06746 1/20 0.52
MAPK1 P28482 1/20 0.46
MAPT P10636 5/20 0.45
TP53 P04637 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.44
GRIN2D O15399 1/20 0.42
GRIN3B O60391 1/20 0.42
GRIN1 Q05586 1/20 0.42
GRIN2A Q12879 1/20 0.42
GRIN2B Q13224 1/20 0.42
GRIN2C Q14957 1/20 0.42
GRIN3A Q8TCU5 1/20 0.42
CYP2C19 P33261 1/20 0.42
ADRB2 P07550 1/20 0.42
ADRB1 P08588 1/20 0.42
ADRB3 P13945 1/20 0.42
GAA P10253 1/20 0.41
HSD11B1 P28845 1/20 0.41
CYP1A2 P05177 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2817033 0.83 ALDH1A1 (0.50) ALDH1A1POLBMAPK1MAPTTP53
SCHEMBL13594836 0.80 ALDH1A1 (0.43) ALDH1A1POLBMAPK1MAPTTP53
SCHEMBL13016868 0.78 GRIN2D (0.47) ALDH1A1MAPTSMN1; SMN2GRIN2DGRIN3B
SCHEMBL396378 0.78 ALDH1A1 (0.46) ALDH1A1POLBMAPK1MAPTTP53
SCHEMBL11176915 0.77 GRIN2D (0.46) ALDH1A1POLBMAPK1MAPTSMN1; SMN2
SCHEMBL7607688 0.77 MAPK1 (0.52) ALDH1A1POLBMAPK1MAPTGAA
SCHEMBL111213 0.76 ALDH1A1 (0.50) ALDH1A1POLBMAPK1MAPTGRIN2D
SCHEMBL428785 0.76 ALDH1A1 (0.49) ALDH1A1POLBMAPK1MAPTHSD11B1
SCHEMBL9190923 0.76 KMT2A (0.42) ALDH1A1POLBMAPK1MAPTTP53
SCHEMBL9265750 0.76 MAPT (0.43) ALDH1A1POLBMAPK1MAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1326606-A2 EP4 RECEPTOR INHIBITORS TO TREAT RHEUMATOID ARTHRITIS PFIZER PHARMACEUTICALS INC. (JP) 2003-07-16 EP disclosed
WO-2002032422-A2 EP4 RECEPTOR INHIBITORS TO TREAT RHEUMATOID ARTHRITIS PFIZER PHARMACEUTICALS INC. (JP) 2002-04-25 WO disclosed