SCHEMBL7019677

SCHEMBL7019677

CCCCc1cccnc1C=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
KAT2B Q92831 1/20 0.35
L3MBTL1 Q9Y468 3/20 0.35
TDP1 Q9NUW8 2/20 0.35
LIPG Q9Y5X9 1/20 0.35
GAA P10253 1/20 0.35
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
TRIM24 O15164 1/20 0.34
TRIM33 Q9UPN9 1/20 0.34
TLR8 Q9NR97 1/20 0.34
GRM5 P41594 1/20 0.34
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
CASP3 P42574 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3800733 0.95 TDP1 (0.41) KAT2BL3MBTL1TDP1LIPGBID
SCHEMBL7857178 0.93 LIPG (0.44) KAT2BL3MBTL1TDP1LIPGBID
SCHEMBL7089971 0.89 GRM5 (0.42) GAATRIM24TRIM33GRM5ALDH1A1
SCHEMBL10968269 0.84 TRIM24 (0.35) L3MBTL1GAATRIM24TRIM33NPC1
SCHEMBL6115316 0.83 TRIM24 (0.39) L3MBTL1TRIM24TRIM33NPC1ALDH1A1
SCHEMBL28102473 0.83 CYP2D6 (0.40) CYP3A4CYP2D6CYP2C9KAT2BL3MBTL1
Benzene SCHEMBL11824212 0.80 TRIM24 (0.37) L3MBTL1GAATRIM24TRIM33NPC1
SCHEMBL3803823 0.79 TRIM24 (0.36) L3MBTL1GAATRIM24TRIM33NPC1
SCHEMBL18995128 0.79 TKT (0.37) L3MBTL1GAATRIM24TRIM33NPC1
SCHEMBL9466495 0.78 THRA (0.41) CYP3A4CYP2D6CYP2C9KAT2BL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101103008-A Macrocyclic compounds useful as bace inhibitors NOVARTIS AG (CH) 2008-01-09 CN disclosed
CN-1535958-A Alpha-substituted pyrimidine. thioalkyl and alkyl ether compound �������Ŷ���Լ��������˾ 2004-10-13 CN disclosed
CN-1152022-C Alpha-substituted pyrimidine-thioalkyl and alkylether compounds �������Ŷ���Լ��������˾ 2004-06-02 CN disclosed
WO-2003084662-A2 COVALENTLY FIXED LIGAND SYSTEMS, NON-METALLOCENE SYSTEMS AND CATALYST SYSTEMS, METHOD FOR THE PRODUCTION THEREOF, AND USE THEREOF FOR POLYMERIZING OLEFINS CELANESE VENTURES GMBH (DE) 2003-10-16 WO disclosed
EP-1317445-A2 CHEMOKINE RECEPTOR BINDING HETEROCYCLIC COMPOUNDS ANORMED INC. (CA) 2003-06-11 EP disclosed
WO-2002022600-A2 CHEMOKINE RECEPTOR BINDING HETEROCYCLIC COMPOUNDS ANORMED INC. (CA) 2002-03-21 WO disclosed
CN-1183773-A Alpha-substituted pyrimidine-thioalkyl and alkylether compounds UPJOHN CO (US) 1998-06-03 CN disclosed
EP-0129791-A2 Tetrahydropyridazinone derivatives, process for their preparation and their use CASSELLA Aktiengesellschaft (DE) 1985-01-02 EP disclosed