SCHEMBL7020146

SCHEMBL7020146

O=c1nc[nH]c2cnsc12

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 2/20 0.32
PARP1 P09874 1/20 0.32
PNP P00491 1/20 0.31
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3417708 0.68 PDPK1 (0.52) PDPK1PARP1ALDH1A1
SCHEMBL3433750 0.62 NPSR1 (0.53) ALDH1A1
SCHEMBL726936 0.61 CNOT7 (0.41) PDPK1PARP1ALDH1A1
SCHEMBL12005970 0.61 LMNA (0.41) PDPK1PNPALDH1A1
SCHEMBL7014722 0.60 PNP (0.34) PDPK1PNPALDH1A1
SCHEMBL1276252 0.60 PDPK1 (0.32) PDPK1PARP1ALDH1A1
SCHEMBL3863547 0.60 CYP1A2 (0.45) PDPK1PARP1ALDH1A1
SCHEMBL6363594 0.59 KDM4C (0.53) PDPK1PARP1ALDH1A1
SCHEMBL3402056 0.59 KDM4C (0.49) PARP1
SCHEMBL15900194 0.59 PNP (0.41) PARP1PNPALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP claimed
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed