SCHEMBL7020883

SCHEMBL7020883

Nc1ncnc2c1c(-c1ccccc1)cn2C1CCCN(OC(=O)O)C1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 11/20 0.67
SRC P12931 10/20 0.67
ABL1 P00519 8/20 0.67
ABL2 P42684 8/20 0.67
BTK Q06187 4/20 0.59
LCK P06239 4/20 0.59
KDR P35968 4/20 0.59
TEK Q02763 3/20 0.59
LYN P07948 2/20 0.59
KDM4E B2RXH2 1/20 0.59
MEN1 O00255 1/20 0.59
RGS12 O14924 1/20 0.59
NPC1 O15118 1/20 0.59
GMNN O75496 1/20 0.59
ALDH1A1 P00352 1/20 0.59
LMNA P02545 1/20 0.59
TP53 P04637 1/20 0.59
CYP1A2 P05177 1/20 0.59
FYN P06241 1/20 0.59
CYP3A4 P08684 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7013342 0.94 SRC (0.67) EGFRSRCABL1ABL2BTK
SCHEMBL27379838 0.90 SRC (0.67) EGFRSRCABL1ABL2BTK
SCHEMBL7021862 0.89 SRC (0.70) EGFRSRCABL1ABL2BTK
SCHEMBL7023217 0.88 SRC (0.71) EGFRSRCABL1ABL2BTK
SCHEMBL7027959 0.86 SRC (0.66) EGFRSRCABL1ABL2KDR
SCHEMBL7019643 0.84 SRC (0.69) EGFRSRCABL1ABL2RIPK2
SCHEMBL28022480 0.84 SRC (0.66) EGFRSRCABL1BTKLCK
SCHEMBL7014659 0.83 ABL1 (0.72) EGFRSRCABL1ABL2LCK
SCHEMBL7023438 0.83 SRC (0.75) EGFRSRCABL1ABL2RIPK2
SCHEMBL8320765 0.82 SRC (0.75) EGFRSRCABL1ABL2BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0888353-B1 N-7-HETEROCYCLYL PYRROLO [2,3-d]PYRIMIDINES AND THEIR USE NOVARTIS AG (CH) 2003-07-09 EP disclosed