SCHEMBL7022256

SCHEMBL7022256

N#Cc1ccc(-c2cc(=O)oc(N)n2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 3/20 0.47
HRH4 Q9H3N8 3/20 0.45
HRH3 Q9Y5N1 2/20 0.45
HTR1A P08908 1/20 0.45
ADRA2A P08913 1/20 0.45
ADRA2C P18825 1/20 0.45
HTR1D P28221 1/20 0.45
HTR2A P28223 1/20 0.45
HTR2C P28335 1/20 0.45
HTR7 P34969 1/20 0.45
MYC P01106 4/20 0.43
NOTUM Q6P988 1/20 0.42
MAOB P27338 2/20 0.40
MAOA P21397 1/20 0.40
XDH P47989 1/20 0.40
CASP1 P29466 1/20 0.40
GAA P10253 1/20 0.40
AR P10275 1/20 0.39
TNKS O95271 1/20 0.38
CA1 P00915 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7261235 0.79 LTA4H (0.46) HRH4NOTUMCA1CA2CA9
SCHEMBL10827533 0.78 ADORA2A (0.52) XDHCA1CA2CA9
SCHEMBL5089384 0.75 TNKS (0.48) PGRMYCNOTUMMAOBMAOA
SCHEMBL29045675 0.73 LTA4H (0.51) HRH4HRH3HTR1AADRA2AADRA2C
SCHEMBL13492147 0.70 ABCG2 (0.57) HRH4HRH3HTR1AADRA2AADRA2C
SCHEMBL20427542 0.69 ADORA1 (0.69) HRH4HRH3HTR1AADRA2AADRA2C
SCHEMBL13288408 0.68 HSP90AA1 (0.62) HRH4HRH3HTR1AADRA2AADRA2C
SCHEMBL31298771 0.68 CFTR (0.45) HRH4HRH3HTR1AADRA2AADRA2C
SCHEMBL19862189 0.67 GAA (0.56) HRH4HRH3HTR1AADRA2AADRA2C
SCHEMBL19868516 0.67 MEN1 (0.55) HRH4HRH3HTR1AADRA2AADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1317433-A2 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2003-06-11 EP disclosed
WO-2002020495-A2 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2002-03-14 WO disclosed
EP-1087963-A1 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 Chiron Corporation (US) 2001-04-04 EP disclosed
WO-1999065897-A1 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 1999-12-23 WO disclosed