SCHEMBL7023745

SCHEMBL7023745

CC(NC(=O)c1ccc2[nH]ccc2c1)C(=O)O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 2/20 0.60
TAS1R1 Q7RTX1 2/20 0.60
PTGS2 P35354 1/20 0.50
MAOA P21397 1/20 0.50
MAOB P27338 1/20 0.50
CTNNB1 P35222 1/20 0.49
WNT3A P56704 1/20 0.49
NPC1 O15118 3/20 0.48
RAB9A P51151 3/20 0.48
MAPT P10636 2/20 0.48
ANPEP P15144 1/20 0.47
CA2 P00918 3/20 0.47
CA1 P00915 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C19 P33261 1/20 0.47
HDAC1 Q13547 2/20 0.46
HDAC2 Q92769 2/20 0.46
HDAC6 Q9UBN7 2/20 0.46
HDAC3 O15379 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8514379 0.87 TAS1R3 (0.68) TAS1R3TAS1R1MAOAMAOBCTNNB1
SCHEMBL14613738 0.80 MAOB (0.47) TAS1R3TAS1R1MAOAMAOBNPC1
SCHEMBL4438920 0.79 MAOA (0.57) TAS1R3TAS1R1MAOAMAOBCTNNB1
SCHEMBL7463164 0.78 TAS1R3 (0.67) TAS1R3TAS1R1MAOAMAOBCTNNB1
Isopropyl Alcohol SCHEMBL28872249 0.77 KDM4E (0.62) TAS1R3TAS1R1PTGS2MAOAMAOB
SCHEMBL9480345 0.77 TAS1R3 (0.60) TAS1R3TAS1R1MAOAMAOBCTNNB1
SCHEMBL1991906 0.77 HDAC6 (0.67) TAS1R3TAS1R1MAOAMAOBCTNNB1
SCHEMBL7463161 0.77 TAS1R3 (0.66) TAS1R3TAS1R1MAOAMAOBCTNNB1
SCHEMBL14121638 0.77 PPARG (0.56) TAS1R3TAS1R1MAOAMAOBCTNNB1
SCHEMBL6706650 0.77 NPC1 (0.54) PTGS2MAOAMAOBNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397360-A1 AZAINDOLES Aventis Pharma Limited (GB) 2004-03-17 EP disclosed
WO-2003000688-A1 AZAINDOLES AVENTIS PHARMA LIMITED (GB) 2003-01-03 WO disclosed