SCHEMBL7025355

SCHEMBL7025355

CCc1ncccc1C(=O)N1CCC(c2cc(O)cc(CN)c2)CC1.c1cc2cc-2c1

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TPSAB1 Q15661 12/20 0.44
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
KCNH2 Q12809 1/20 0.40
F10 P00742 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4403358 0.99 TPSAB1 (0.43) TPSAB1CYP3A4CYP2D6KCNH2F10
Hydrochloric Acid SCHEMBL4404473 0.89 TPSAB1 (0.54) TPSAB1CYP3A4CYP2D6KCNH2F10
Hydrochloric Acid SCHEMBL6491184 0.87 TPSAB1 (0.43) TPSAB1CYP3A4CYP2D6KCNH2
SCHEMBL7019482 0.84 TPSAB1 (0.40) TPSAB1CYP3A4CYP2D6KCNH2F10
Hydrochloric Acid SCHEMBL4404747 0.83 TPSAB1 (0.40) TPSAB1CYP3A4CYP2D6KCNH2F10
SCHEMBL4399231 0.82 TPSAB1 (0.40) TPSAB1CYP3A4CYP2D6KCNH2F10
Hydrochloric Acid SCHEMBL4401946 0.81 TPSAB1 (0.40) TPSAB1CYP3A4CYP2D6KCNH2F10
SCHEMBL4412828 0.81 TPSAB1 (0.49) TPSAB1CYP3A4CYP2D6KCNH2F10
Hydrochloric Acid SCHEMBL4406550 0.81 HTR2A (0.39) TPSAB1
Hydrochloric Acid SCHEMBL4414531 0.81 TPSAB1 (0.49) TPSAB1CYP3A4CYP2D6KCNH2F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1296972-A1 ARYLMETHYLAMINE DERIVATIVES FOR USE AS TRYPTASE INHIBITORS Aventis Pharmaceuticals Inc. (US) 2003-04-02 EP disclosed
WO-2001090101-A1 ARYLMETHYLAMINE DERIVATIVES FOR USE AS TRYPTASE INHIBITORS AVENTIS PHARMACEUTICALS INC. (US) 2001-11-29 WO disclosed