SCHEMBL7029182

SCHEMBL7029182

Nc1nnc(-c2ccccc2)c(=O)n1N

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 8/20 0.44
ADORA2A P29274 4/20 0.44
ADORA2B P29275 5/20 0.44
KMT2A Q03164 2/20 0.44
CSNK1A1 P48729 2/20 0.43
CLK4 Q9HAZ1 2/20 0.43
ADORA3 P0DMS8 2/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
FGFR1 P11362 2/20 0.39
FLT1 P17948 2/20 0.39
KDR P35968 2/20 0.39
CSF1R P07333 1/20 0.39
CDK8 P49336 1/20 0.39
GSK3A P49840 1/20 0.39
GSK3B P49841 1/20 0.39
CDK5 Q00535 1/20 0.39
PRKCQ Q04759 1/20 0.39
LRRK2 Q5S007 1/20 0.39
DYRK1B Q9Y463 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11722694 0.82 ADORA1 (0.44) ADORA1ADORA2AADORA2BKMT2AADORA3
SCHEMBL11717758 0.80 ADORA1 (0.43) ADORA1ADORA2AADORA2BKMT2ACSNK1A1
Metamitron SCHEMBL66369 0.80 KDM4E (0.49) ADORA1ADORA2BKMT2AADORA3NPC1
Metamitron SCHEMBL8536394 0.80 KDM4E (0.49) ADORA1ADORA2BKMT2AADORA3NPC1
SCHEMBL11064095 0.80 ADORA1 (0.54) ADORA1ADORA2AADORA2BCSNK1A1CLK4
SCHEMBL11385843 0.80 ADORA1 (0.43) ADORA1ADORA2AADORA2BKMT2ACSNK1A1
SCHEMBL11602304 0.76 ALDH1A1 (0.49) ADORA1ADORA2BKMT2AADORA3KDM4E
SCHEMBL10508760 0.76 ALDH1A1 (0.61) ADORA1ADORA2BKMT2ACSNK1A1CLK4
SCHEMBL11609509 0.76 ALDH1A1 (0.48) ADORA1ADORA2AADORA2BKMT2ANPC1
SCHEMBL11715949 0.76 ADORA1 (0.43) ADORA1ADORA2AADORA2BKMT2AADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889884-B1 1,2,4-TRIAZINE DERIVATIVES FOR THE INHIBITION OF PROTEIN GLYCOSYLATION ALTEON INC (US) 2003-01-29 EP disclosed
US-4036632-A CONTROLLING WEEDS USING 3-METHYLTHIO-4-AMINO-6-BUTYL-1,2,4 TRIAZINE-5-ONE BAYER AKTIENGESELLSCHAFT (DT) 1977-07-19 US disclosed
US-3966715-A 1,2,4-TRIAZINE-5-ONES BAYER AKTIENGESELLSCHAFT (DT) 1976-06-29 US disclosed
US-3961936-A SUBSTITUTED 1,2,4-TRIAZINE-5-ONES BAYER AKTIENGESELLSCHAFT (DT) 1976-06-08 US disclosed