SCHEMBL11064095

SCHEMBL11064095

Cn1c(N)nnc(-c2ccccc2)c1=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 6/20 0.54
ADORA2B P29275 3/20 0.54
ALDH1A1 P00352 4/20 0.50
KDM4E B2RXH2 3/20 0.50
GAA P10253 2/20 0.50
HPGD P15428 2/20 0.50
CLK4 Q9HAZ1 3/20 0.44
CSNK1A1 P48729 2/20 0.44
CDK8 P49336 2/20 0.44
CSF1R P07333 1/20 0.44
FGFR1 P11362 1/20 0.44
FLT1 P17948 1/20 0.44
KDR P35968 1/20 0.44
GSK3A P49840 1/20 0.44
GSK3B P49841 1/20 0.44
CDK5 Q00535 1/20 0.44
PRKCQ Q04759 1/20 0.44
LRRK2 Q5S007 1/20 0.44
DYRK1B Q9Y463 1/20 0.44
CYP1A2 P05177 4/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7029182 0.80 ADORA1 (0.44) ADORA1ADORA2BALDH1A1KDM4EHPGD
SCHEMBL9843278 0.76 ADORA1 (0.51) ADORA1ADORA2BALDH1A1KDM4EGAA
SCHEMBL10841723 0.76 KDM4E (0.54) ADORA1ADORA2BALDH1A1KDM4EGAA
SCHEMBL11813567 0.76 ADORA2B (0.51) ADORA1ADORA2BALDH1A1KDM4EGAA
SCHEMBL11808587 0.76 ADORA1 (0.51) ADORA1ADORA2BALDH1A1KDM4EGAA
SCHEMBL10843009 0.75 KDM4E (0.53) ADORA1ADORA2BALDH1A1KDM4EGAA
SCHEMBL13872765 0.73 KMT2A (0.54) ADORA1ADORA2BALDH1A1CYP1A2CYP3A4
Metamitron SCHEMBL8536394 0.71 KDM4E (0.49) ADORA1ADORA2BALDH1A1KDM4EGAA
Metamitron SCHEMBL66369 0.71 KDM4E (0.49) ADORA1ADORA2BALDH1A1KDM4EGAA
SCHEMBL11609509 0.68 ALDH1A1 (0.48) ADORA1ADORA2BALDH1A1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4447258-A 3-Dimethylamino-4-methyl-1,2,4-triazin-5(4H)-ones and herbicidal compositions BAYER AKTIENGESELLSCHAFT (DE) 1984-05-08 US disclosed
EP-0015452-B1 6-SUBSTITUTED-3-DIMETHYLAMINO-4-METHYL-1,2,4-TRIAZIN-5-(4H)-ONES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS HERBICIDES BAYER AG (DE) 1982-01-20 EP disclosed
EP-0015452-A1 6-Substituted-3-dimethylamino-4-methyl-1,2,4-triazin-5-(4H)-ones, processes for their preparation and their use as herbicides BAYER AG (DE) 1980-09-17 EP disclosed