SCHEMBL7029249

SCHEMBL7029249

CCCCCC(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)/C=C(\C)C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CES2 O00748 4/20 0.37
LPAR1 Q92633 1/20 0.33
LPAR3 Q9UBY5 1/20 0.33
FAAH O00519 9/20 0.33
CES1 P23141 5/20 0.32
MEN1 O00255 1/20 0.32
CYP1A2 P05177 1/20 0.32
KMT2A Q03164 1/20 0.32
HSD17B10 Q99714 1/20 0.32
EP300 Q09472 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7029253 1.00 CES2 (0.37) CES2LPAR1LPAR3FAAHCES1
SCHEMBL1769903 0.94 CES2 (0.32) CES2FAAHCES1MEN1CYP1A2
SCHEMBL848224 0.83
SCHEMBL2680481 0.83
SCHEMBL8520645 0.83
SCHEMBL1581509 0.82
SCHEMBL1581276 0.82
SCHEMBL1581563 0.82
SCHEMBL14861335 0.82
SCHEMBL1581124 0.82

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1280929-A2 VECTORS FOR OCULAR TRANSDUCTION AND USE THEREOF FOR GENETIC THERAPY Novartis AG (CH) 2003-02-05 EP disclosed
WO-2001083729-A2 VECTORS FOR OCULAR TRANSDUCTION AND USE THEREOF FOR GENETIC THERAPY NOVARTIS AG (CH) 2001-11-08 WO disclosed
EP-1082142-A2 COMPOSITIONS AND METHODS FOR DELIVERY OF GENETIC MATERIAL FOR ALTERING NEURONAL GROWTH, REGENERATION, AND SURVIVAL Selective Genetics, Inc. (US) 2001-03-14 EP disclosed
WO-1999066959-A9 COMPOSITIONS AND METHODS FOR DELIVERY OF GENETIC MATERIAL FOR ALTERING NEURONAL GROWTH, REGENERATION, AND SURVIVAL SELECTIVE GENETICS INC (US) 2000-03-30 WO disclosed
EP-0973926-A1 ADENOVIRAL VECTORS WITH MODIFIED TROPISM Selective Genetics, Inc. (US) 2000-01-26 EP disclosed
WO-1999066959-A2 COMPOSITIONS AND METHODS FOR DELIVERY OF GENETIC MATERIAL FOR ALTERING NEURONAL GROWTH, REGENERATION, AND SURVIVAL SELECTIVE GENETICS, INC. (US) 1999-12-29 WO disclosed
WO-1998040508-A1 ADENOVIRAL VECTORS WITH MODIFIED TROPISM SELECTIVE GENETICS, INC. (US) 1998-09-17 WO disclosed
WO-1998039436-A2 FIBROBLAST GROWTH FACTOR MUTEIN COMPOSITIONS AND METHODS OF USE THEREFOR EISAI CO., LTD. (JP) 1998-09-11 WO disclosed
EP-0833665-A1 COMPOSITIONS CONTAINING NUCLEIC ACIDS AND LIGANDS FOR THERAPEUTIC TREATMENT PRIZM PHARMACEUTICALS, INC. (US) 1998-04-08 EP disclosed
EP-0776218-A2 HEPARIN-BINDING GROWTH FACTORS FOR GENE THERAPY AND ANTERIOR EYE DISORDERS PRIZM PHARMACEUTICALS, INC. (US) 1997-06-04 EP disclosed
EP-0754046-A1 USE OF PHOSPHONYLMETHOXYALKYL NUCLEOSIDES FOR THE TREATMENT OF RAISED INTRAOCULAR PRESSURE FREEMAN, William R. (US) 1997-01-22 EP disclosed
WO-1996036362-A1 COMPOSITIONS CONTAINING NUCLEIC ACIDS AND LIGANDS FOR THERAPEUTIC TREATMENT PRIZM PHARMACEUTICALS, INC. (US) 1996-11-21 WO disclosed
WO-1995026734-A1 USE OF PHOSPHONYLMETHOXYALKYL NUCLEOSIDES FOR THE TREATMENT OF RAISED INTRAOCULAR PRESSURE FREEMAN WILLIAM R (US) 1995-10-12 WO disclosed
WO-1995024928-A2 HEPARIN-BINDING GROWTH FACTORS FOR GENE THERAPY AND ANTERIOR EYE DISORDERS PRIZM PHARMACEUTICALS, INC. (US) 1995-09-21 WO disclosed