SCHEMBL7030152

SCHEMBL7030152

CCCn1c(-c2ccccc2)nc2c1c(=O)n(C)c(=O)n2C

nearest known ligand 0.70

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 6/20 0.70
ADORA2A P29274 2/20 0.70
LMNA P02545 3/20 0.60
TSHR P16473 2/20 0.60
HTT P42858 2/20 0.60
NPSR1 Q6W5P4 1/20 0.60
SMN1; SMN2 Q16637 2/20 0.59
JAK2 O60674 1/20 0.59
HPGD P15428 1/20 0.56
ALDH1A1 P00352 1/20 0.54
GAA P10253 1/20 0.54
USP2 O75604 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL683962 0.86 ADORA2B (0.62) ADORA2BADORA2ALMNATSHRHTT
SCHEMBL7037369 0.86 ADORA2B (0.88) ADORA2BADORA2AALDH1A1
Hydrochloric Acid SCHEMBL11388923 0.85 ADORA2B (0.61) ADORA2BADORA2ALMNATSHRHTT
Diethylamine SCHEMBL11388706 0.85 ADORA2B (0.64) ADORA2BADORA2ALMNATSHRSMN1; SMN2
SCHEMBL17626266 0.84 ADORA2B (0.67) ADORA2BADORA2ALMNATSHRSMN1; SMN2
Diethylamine SCHEMBL11388925 0.84 ADORA2B (0.62) ADORA2BADORA2ALMNATSHRSMN1; SMN2
SCHEMBL8318291 0.83 ADORA2B (0.58) ADORA2BADORA2ALMNATSHRHTT
SCHEMBL4146728 0.83 ADORA2B (1.00) ADORA2BADORA2AHTTSMN1; SMN2HPGD
SCHEMBL10395302 0.81 ADORA2B (0.63) ADORA2BADORA2AHPGDALDH1A1
SCHEMBL515794 0.78 ADORA2B (0.74) ADORA2BADORA2AHTTSMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0956855-B1 Immunosuppressive effects of 8 substituted xanthine derivatives LEUVEN K U RES & DEV (BE) 2003-03-12 EP claimed