SCHEMBL8318291

SCHEMBL8318291

CCN(CO)CCn1c(-c2ccccc2)nc2c1c(=O)n(C)c(=O)n2C

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 6/20 0.58
ADORA2A P29274 2/20 0.58
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
TSHR P16473 3/20 0.49
LMNA P02545 2/20 0.49
NPSR1 Q6W5P4 2/20 0.49
HTT P42858 1/20 0.49
HPGD P15428 1/20 0.48
TP53 P04637 1/20 0.48
MAPT P10636 1/20 0.48
MAOB P27338 1/20 0.47
ALDH1A1 P00352 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL683962 0.94 ADORA2B (0.62) ADORA2BADORA2AMEN1KMT2ATSHR
Hydrochloric Acid SCHEMBL11388923 0.93 ADORA2B (0.61) ADORA2BADORA2AMEN1KMT2ATSHR
SCHEMBL683888 0.85 SMN1; SMN2 (0.51) ADORA2BADORA2AMEN1KMT2ATSHR
Hydrochloric Acid SCHEMBL11381649 0.84 SMN1; SMN2 (0.50) ADORA2BADORA2AMEN1KMT2ATSHR
SCHEMBL7030152 0.83 ADORA2B (0.70) ADORA2BADORA2ATSHRLMNANPSR1
SCHEMBL684271 0.83 TSHR (0.54) ADORA2BADORA2AMEN1KMT2ATSHR
Hydrochloric Acid SCHEMBL11384998 0.82 TSHR (0.53) ADORA2BADORA2AMEN1KMT2ATSHR
SCHEMBL683542 0.81 NCOA3 (0.54) ADORA2BADORA2AMEN1KMT2ATSHR
Hydrochloric Acid SCHEMBL11381068 0.81 NCOA3 (0.53) ADORA2BADORA2AMEN1KMT2ATSHR
SCHEMBL682765 0.81 MAOB (0.49) ADORA2BADORA2ATP53MAOBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004067006-A1 COMBINATION OF A PDE IV INHIBITOR AND A TNF-ALPHA ANTAGONIST PHARMACIA CORPORATION (US) 2004-08-12 WO disclosed