SCHEMBL7030588

SCHEMBL7030588

O=C(O)N1CCc2c(n3c4c(cccc24)CCC3)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 4/20 0.52
KDM4E B2RXH2 4/20 0.49
HSD17B10 Q99714 4/20 0.49
CYP1A2 P05177 2/20 0.49
LMNA P02545 1/20 0.49
HTR2C P28335 4/20 0.46
HTR2A P28223 3/20 0.46
KMT2A Q03164 3/20 0.46
MEN1 O00255 2/20 0.46
TP53 P04637 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
MAPT P10636 1/20 0.46
CYP2C9 P11712 1/20 0.46
ALOX15 P16050 1/20 0.46
MAPK1 P28482 1/20 0.46
CYP2C19 P33261 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
ALDH1A1 P00352 2/20 0.45
USP2 O75604 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6493920 0.81 PTGDR2 (0.50) KDM4EHSD17B10CYP1A2LMNAHTR2C
SCHEMBL6485143 0.80 HTR2C (0.46) MCL1KDM4EHSD17B10CYP1A2LMNA
SCHEMBL3545060 0.80 HTR2C (0.67) MCL1KDM4EHSD17B10CYP1A2LMNA
SCHEMBL7038582 0.80 HTR2C (0.48) MCL1KDM4EHSD17B10LMNAHTR2C
SCHEMBL7034581 0.80 PTGDR2 (0.38) MCL1KDM4EHSD17B10CYP1A2HTR2C
SCHEMBL3550600 0.79 HTR2C (0.68) MCL1KDM4EHSD17B10CYP1A2LMNA
SCHEMBL6850296 0.77 PDE3B (0.38) MCL1KDM4EHTR2CHTR2AKMT2A
SCHEMBL5413796 0.75 HTR2C (0.60) MCL1KDM4EHSD17B10CYP1A2LMNA
SCHEMBL6491761 0.75 CHRM1 (0.38) MCL1HTR2CHTR2A
SCHEMBL6496372 0.75 PTGDR2 (0.36) KDM4EHSD17B10CYP1A2HTR2CHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1173440-B1 TETRACYCLIC AZEPINOINDOLE COMPOUNDS AS 5-HT RECEPTOR LIGANDS UPJOHN CO (US) 2004-09-15 EP claimed