SCHEMBL6850296

SCHEMBL6850296

O=C(O)N1CCc2c(n3c4c(ccc(Cc5ccccc5)c24)CCC3)CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38
ALDH1A1 P00352 2/20 0.37
HTT P42858 1/20 0.37
LIPG Q9Y5X9 2/20 0.36
ALOX5 P09917 2/20 0.36
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
MCL1 Q07820 2/20 0.34
HSP90AA1 P07900 1/20 0.34
TDP1 Q9NUW8 2/20 0.34
RORC P51449 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
RECQL P46063 1/20 0.34
CACNA1B Q00975 1/20 0.33
KDM4E B2RXH2 1/20 0.32
PTGS1 P23219 1/20 0.32
NQO1 P15559 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7030588 0.77 MCL1 (0.52) ALDH1A1HTTLIPGHTR2AHTR2C
SCHEMBL6497695 0.70 ALDH1A1 (0.45) ALDH1A1HTR2AMEN1KMT2AKDM4E
SCHEMBL7038582 0.65 HTR2C (0.48) ALDH1A1HTR2AHTR2CMCL1TDP1
SCHEMBL7034581 0.65 PTGDR2 (0.38) ALDH1A1LIPGHTR2AHTR2CMCL1
SCHEMBL6492932 0.63 MEN1 (0.46) MEN1KMT2A
SCHEMBL6493228 0.63 PTGDR2 (0.47) MEN1KMT2A
SCHEMBL6850299 0.61 KDM4E (0.38) HTR2BTDP1MEN1KMT2AKDM4E
SCHEMBL7680290 0.61 NOTUM (0.33) MCL1
SCHEMBL7676778 0.60 HTR2C (0.37) ALDH1A1HTR2AHTR2CMCL1
SCHEMBL7679724 0.60 HTR2A (0.36) HTR2AHTR2CMCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1173440-B1 TETRACYCLIC AZEPINOINDOLE COMPOUNDS AS 5-HT RECEPTOR LIGANDS UPJOHN CO (US) 2004-09-15 EP claimed