SCHEMBL7030804

SCHEMBL7030804

CN1CCN(c2cccc3c2CC[C@H](N(Cc2ccccc2)Cc2ccccc2)C3)CC1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 15/20 0.56
DRD3 P35462 11/20 0.56
DRD1 P21728 4/20 0.49
DRD4 P21917 3/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
TSHR P16473 1/20 0.49
NFKB1 P19838 1/20 0.49
THPO P40225 1/20 0.49
LMNA P02545 1/20 0.48
PMP22 Q01453 1/20 0.48
HTR1A P08908 3/20 0.48
HTR7 P34969 3/20 0.48
DRD5 P21918 1/20 0.45
ADRB2 P07550 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7025402 1.00 DRD2 (0.56) DRD2DRD3DRD1DRD4CYP1A2
SCHEMBL6816670 0.91 DRD2 (0.48) DRD2DRD3
SCHEMBL7030108 0.91 DRD2 (0.48) DRD2DRD3
SCHEMBL8157601 0.91 DRD2 (0.48) DRD2DRD3
SCHEMBL7239524 0.84 DRD2 (0.43) DRD2DRD3
SCHEMBL7027796 0.83 DRD2 (0.51) DRD2DRD3DRD1DRD4CYP1A2
SCHEMBL7025218 0.83 DRD2 (0.51) DRD2DRD3DRD1DRD4CYP1A2
SCHEMBL7020675 0.83 DRD2 (0.52) DRD2DRD3
SCHEMBL6819394 0.83 DRD2 (0.43) DRD2DRD3DRD1CYP1A2CYP3A4
SCHEMBL7244550 0.83 DRD2 (0.46) DRD2DRD3DRD1DRD4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0888319-B1 SUBSTITUTED 1,2,3,4-TETRAHYDRONAPHTHALENE DERIVATIVES ASTRAZENECA AB (SE) 2003-01-29 EP disclosed
US-6410530-B1 CENTRAL NERVOUS SYSTEM DISORDERS; PSYCHOLOGICAL DISORDERS ASTRAZENECA AB (SE) 2002-06-25 US disclosed
US-6124283-A Substituted 1,2,3,4-tetrahydronaphthalene derivatives ASTRA AKTIEBOLAG (SE) 2000-09-26 US disclosed