SCHEMBL7033409

SCHEMBL7033409

C=CCc1ccc2[nH]c(=O)[nH]c(=O)c2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.46
CA9 Q16790 2/20 0.46
KDM4E B2RXH2 8/20 0.44
PARP1 P09874 2/20 0.44
GAA P10253 4/20 0.40
PKM P14618 1/20 0.40
XDH P47989 1/20 0.40
ALDH1A1 P00352 6/20 0.39
HPGD P15428 3/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
KMT2A Q03164 4/20 0.39
MAPT P10636 4/20 0.39
MEN1 O00255 3/20 0.39
PPARG P37231 2/20 0.39
PPARD Q03181 2/20 0.39
ALDH2 P05091 1/20 0.39
GABRA1 P14867 1/20 0.39
AKR1B1 P15121 1/20 0.39
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7030477 0.87 PARP1 (0.44) CA12CA9KDM4EPARP1GAA
SCHEMBL24451736 0.81 ALDH1A1 (0.48) KDM4EPARP1GAAXDHALDH1A1
SCHEMBL7028337 0.78 CA12 (0.50) CA12CA9KDM4EPARP1GAA
SCHEMBL2056368 0.78 ALDH1A1 (0.50) CA12CA9KDM4EPARP1GAA
SCHEMBL7034143 0.78 CA12 (0.50) CA12CA9KDM4EPARP1GAA
SCHEMBL20942693 0.78 GAA (0.66) CA12CA9KDM4EPARP1GAA
SCHEMBL7028562 0.75 CA12 (0.47) CA12CA9KDM4EPARP1GAA
SCHEMBL7033620 0.75 CA12 (0.47) CA12CA9KDM4EPARP1GAA
SCHEMBL7030539 0.75 CA12 (0.50) CA12CA9KDM4EPARP1ALDH1A1
SCHEMBL7028533 0.74 KDM4E (0.53) CA12CA9KDM4EPARP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0878468-B1 Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL CO (JP) 2003-03-19 EP disclosed
EP-0775697-B1 Process for producing 1-substituted tetrahydroquinazolindionen SUMITOMO CHEMICAL CO (JP) 2003-02-12 EP disclosed
US-5994542-A Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1999-11-30 US disclosed
EP-0878468-A1 Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-11-18 EP disclosed
US-5756738-A Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-05-26 US disclosed
EP-0775697-A1 Process for producing 1-substituted tetrahydroquinazolindionen SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-05-28 EP disclosed