SCHEMBL7034353

SCHEMBL7034353

O=c1[nH]c(=O)c2ccc(Cl)c(Br)c2[nH]1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.40
CSNK2A2 P19784 1/20 0.40
CSNK2B P67870 1/20 0.40
CSNK2A1 P68400 1/20 0.40
DAO P14920 2/20 0.39
PARP1 P09874 2/20 0.37
KDM4E B2RXH2 1/20 0.37
CA12 O43570 1/20 0.37
CA9 Q16790 1/20 0.37
TYMP P19971 8/20 0.36
GSK3B P49841 1/20 0.36
BACE1 P56817 1/20 0.36
PNP P00491 1/20 0.35
GDA Q9Y2T3 1/20 0.34
MAPT P10636 1/20 0.34
XDH P47989 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7032317 0.81 PARP1 (0.37) IDH1CSNK2A2CSNK2BCSNK2A1DAO
SCHEMBL7032941 0.81 IDH1 (0.43) IDH1CSNK2A2CSNK2BCSNK2A1DAO
SCHEMBL3671768 0.81 CSNK2A2 (0.41) CSNK2A2CSNK2BCSNK2A1DAOPARP1
SCHEMBL27299278 0.78 PARP1 (0.37) DAOPARP1KDM4ECA12CA9
SCHEMBL27296153 0.74 ALDH1A1 (0.40) DAOPARP1KDM4ECA12CA9
SCHEMBL2922284 0.73 DAO (0.60) DAOPARP1KDM4ECA12CA9
SCHEMBL25988754 0.73 IDH1 (0.39) IDH1CSNK2A2CSNK2BCSNK2A1DAO
SCHEMBL23540965 0.71 AR (0.41) IDH1CSNK2A2CSNK2BCSNK2A1DAO
SCHEMBL29947950 0.71 AR (0.41) IDH1CSNK2A2CSNK2BCSNK2A1DAO
SCHEMBL25601009 0.71 IDH1 (0.38) IDH1CSNK2A2CSNK2BCSNK2A1DAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0878468-B1 Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL CO (JP) 2003-03-19 EP disclosed
EP-0775697-B1 Process for producing 1-substituted tetrahydroquinazolindionen SUMITOMO CHEMICAL CO (JP) 2003-02-12 EP disclosed
US-5994542-A Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1999-11-30 US disclosed
EP-0878468-A1 Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-11-18 EP disclosed
US-5756738-A Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-05-26 US disclosed
EP-0775697-A1 Process for producing 1-substituted tetrahydroquinazolindionen SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-05-28 EP disclosed