SCHEMBL7036293

SCHEMBL7036293

CC1CNc2cc(N)ccc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.42
CHRNA4 P43681 1/20 0.42
KDM4E B2RXH2 2/20 0.38
MEN1 O00255 2/20 0.38
GAA P10253 2/20 0.38
MAPT P10636 2/20 0.38
KMT2A Q03164 2/20 0.38
APAF1 O14727 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
AR P10275 1/20 0.36
CA9 Q16790 2/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
HTR2C P28335 7/20 0.33
HTR2A P28223 6/20 0.33
HTR2B P41595 5/20 0.33
ALDH1A1 P00352 2/20 0.31
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6650256 0.81 AR (0.39) CHRNB2CHRNA4KDM4EMEN1GAA
SCHEMBL12413 0.78 CA1 (0.45) CHRNB2CHRNA4GAAMAPTKMT2A
SCHEMBL13894872 0.77 HTR2C (0.51) CHRNB2CHRNA4GAAARCA1
SCHEMBL31158608 0.77 HTR2C (0.49) CHRNB2CHRNA4MEN1KMT2AAR
SCHEMBL13168986 0.77 CHRNB2 (0.39) CHRNB2CHRNA4KDM4EMEN1GAA
SCHEMBL8180143 0.75 MKNK1 (0.44) CHRNB2CHRNA4TDP1CA9CA12
SCHEMBL8178575 0.75 MKNK1 (0.44) CHRNB2CHRNA4TDP1CA9CA12
SCHEMBL6651725 0.74 KDM4E (0.39) CHRNB2CHRNA4KDM4EMEN1GAA
SCHEMBL8081529 0.74 ESR2 (0.35) ARHTR2CHTR2AHTR2B
SCHEMBL12983195 0.74 PARP1 (0.37) KDM4EGAAARHTR2CHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 43 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0575604-B2 INDOLINE PRODUCTS, METHODS FOR PREPARING SAME, AND USE THEREOF IN COSMETICS OREAL (FR) 2003-03-26 EP claimed
US-5776497-A OXIDATIVE POLYMERIZATION OF INDOLINE FOR COSMETICS L'OREAL (FR) 1998-07-07 US claimed
EP-0544874-B1 METHOD FOR PREPARING SUBMICRON PARTICLES IN THE PRESENCE OF LIPID VESICLES, AND CORRESPONDING COMPOSITIONS OREAL (FR) 1998-04-08 EP claimed
US-5670099-A PREPARING A DISPERSION OF LIPIDIC VESICLES FROM ATLEAST ONE LIPID, AN AQUEOUS PHASE ENCAPSULATED IN VESICLE, DISSOLVING POLYMERIZABLE INDOLIC OR INDOLINIC MONOMER WITH A POLYMERIZATION AGENT, REACTS WITH MONOMER FORMS PARTICLES L'OREAL (FR) 1997-09-23 US claimed
US-5583234-A Indoline-based products, processes for preparing them and their use in cosmetics L'OREAL (FR) 1996-12-10 US claimed
EP-0575605-B1 MINERAL OR ORGANIC PARTICLE BASED PRODUCT COMPRISING AN INDOLINE PRODUCT OREAL (FR) 1996-11-27 EP claimed
US-5496543-A COSMETICS L'OREAL (FR) 1996-03-05 US claimed
EP-0575604-B1 INDOLINE PRODUCTS, METHODS FOR PREPARING SAME, AND USE THEREOF IN COSMETICS OREAL (FR) 1995-12-06 EP claimed
EP-0575605-A1 MINERAL OR ORGANIC PARTICLE BASED PRODUCT COMPRISING AN INDOLINE PRODUCT. OREAL (FR) 1993-12-29 EP claimed
EP-0575604-A1 INDOLINE PRODUCTS, METHODS FOR PREPARING SAME, AND USE THEREOF IN COSMETICS. OREAL (FR) 1993-12-29 EP claimed
WO-1993013744-A1 INDOLINE PRODUCTS, METHODS FOR PREPARING SAME, AND USE THEREOF IN COSMETICS L'OREAL (FR) 1993-07-22 WO claimed
WO-1993013745-A1 MINERAL OR ORGANIC PARTICLE BASED PRODUCT COMPRISING AN INDOLINE PRODUCT L'OREAL (FR) 1993-07-22 WO claimed
EP-0544874-A1 METHOD FOR PREPARING SUBMICRON PARTICLES IN THE PRESENCE OF LIPID VESICLES, AND CORRESPONDING COMPOSITIONS L'OREAL (FR) 1993-06-09 EP claimed
WO-1993000068-A1 METHOD FOR PREPARING SUBMICRON PARTICLES IN THE PRESENCE OF LIPID VESICLES, AND CORRESPONDING COMPOSITIONS L'OREAL (FR) 1993-01-07 WO claimed
EP-0575604-B2 INDOLINE PRODUCTS, METHODS FOR PREPARING SAME, AND USE THEREOF IN COSMETICS OREAL (FR) 2003-03-26 EP disclosed
WO-2002102333-A1 COATED ORGANIC PIGMENT AND COSMETIC COMPOSITION CONTAINING SAID PIGMENT L'OREAL (FR) 2002-12-27 WO disclosed
US-6432417-B1 CONTAINING PRIMARY, SECONDARY, TERTIARY AND/OR QUATERNARY AMINE GROUPINGS; READILY DISPERSIBLE, EVEN IN FATTY BINDERS L'OREAL (FR) 2002-08-13 US disclosed
WO-1993013744-A1 INDOLINE PRODUCTS, METHODS FOR PREPARING SAME, AND USE THEREOF IN COSMETICS L'OREAL (FR) 1993-07-22 WO disclosed
EP-0544874-A1 METHOD FOR PREPARING SUBMICRON PARTICLES IN THE PRESENCE OF LIPID VESICLES, AND CORRESPONDING COMPOSITIONS L'OREAL (FR) 1993-06-09 EP disclosed
WO-1993000068-A1 METHOD FOR PREPARING SUBMICRON PARTICLES IN THE PRESENCE OF LIPID VESICLES, AND CORRESPONDING COMPOSITIONS L'OREAL (FR) 1993-01-07 WO disclosed