SCHEMBL7036876

SCHEMBL7036876

CCn1nc(-c2cccc(O)c2)ccc1=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 4/20 0.51
ADORA2A P29274 2/20 0.51
ADORA2B P29275 2/20 0.51
ADORA1 P30542 2/20 0.51
GABRA1 P14867 1/20 0.50
GABRB2 P47870 1/20 0.50
USP2 O75604 1/20 0.49
PKM P14618 1/20 0.49
ALOX15 P16050 1/20 0.49
ATM Q13315 1/20 0.49
HTT P42858 1/20 0.48
FYN P06241 3/20 0.46
HSD17B1 P14061 2/20 0.44
HSD17B2 P37059 2/20 0.44
MET P08581 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HSD17B10 Q99714 1/20 0.43
KDM4E B2RXH2 1/20 0.42
PDE4A P27815 1/20 0.42
PDE4C Q08493 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7035765 0.89 GABRA1 (0.51) PDE4BADORA2AADORA2BADORA1GABRA1
SCHEMBL15317761 0.85 GABRA1 (0.47) PDE4BADORA2AADORA2BADORA1GABRA1
SCHEMBL4054250 0.82 KDM4E (0.55) PDE4BHTTMETKDM4EPDE4A
SCHEMBL8866625 0.82 GABRA1 (0.47) PDE4BADORA2AADORA2BADORA1GABRA1
SCHEMBL10194702 0.81 KDM4E (0.52) GABRA1GABRB2HTTSMN1; SMN2HSD17B10
SCHEMBL4054492 0.81 HTT (0.62) HTTSMN1; SMN2HSD17B10KDM4EMEN1
SCHEMBL2823853 0.80 MEN1 (0.53) PDE4BHTTMETSMN1; SMN2PDE4A
Bromide SCHEMBL5751833 0.80 HTT (0.61) HTTSMN1; SMN2HSD17B10KDM4EMEN1
SCHEMBL7037096 0.79 KDM4E (0.51) PDE4BHTTMETSMN1; SMN2HSD17B10
SCHEMBL14494768 0.78 MET (0.50) PDE4BMETSMN1; SMN2PDE4APDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2655357-B1 INDAZOLYL TRIAZOLE DERIVATIVES AS IRAK INHIBITORS MERCK SERONO SA (CH) 2016-06-22 EP disclosed
WO-2012084704-A1 INDAZOLYL TRIAZOLE DERIVATIVES AS IRAK INHIBITORS MERCK SERONO S.A. (CH) 2012-06-28 WO disclosed
EP-0835865-B1 Dihydropyridazinones and pyridazinones and their use as fungicides and insecticides DOW AGROSCIENCES LLC (US) 2003-03-12 EP disclosed
US-6121251-A CONTROLLING PHYTOPATHOGENIC FUNGI, INSECTS ROHM AND HAAS COMPANY (US) 2000-09-19 US disclosed
EP-0835865-A1 Dihydropyridazinones and pyridazinones and their use as fungicides and insecticides ROHM AND HAAS COMPANY (US) 1998-04-15 EP disclosed