SCHEMBL7040485

SCHEMBL7040485

COc1cc2c(cc1C=O)C(Cc1c[nH]cn1)CC2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.39
NQO2 P16083 2/20 0.38
MTNR1A P48039 2/20 0.38
MTNR1B P49286 2/20 0.38
ALDH1A1 P00352 3/20 0.37
GAA P10253 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
KDM4E B2RXH2 1/20 0.35
TSHR P16473 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
POLA1 P09884 2/20 0.35
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
LMNA P02545 1/20 0.33
HPGD P15428 1/20 0.33
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32
PPARD Q03181 3/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7038086 0.96 NQO2 (0.38) ESR1NQO2MTNR1AMTNR1BALDH1A1
SCHEMBL7038524 0.87 NQO2 (0.46) NQO2MTNR1AMTNR1BALDH1A1KDM4E
SCHEMBL7035810 0.83 ADRA2A (0.39) ESR1POLA1
SCHEMBL7037840 0.82 NQO2 (0.37) NQO2MTNR1AMTNR1BALDH1A1KDM4E
SCHEMBL7038059 0.81 NQO2 (0.46) NQO2MTNR1AMTNR1BALDH1A1KDM4E
SCHEMBL7035027 0.81 ADRA2A (0.39) ESR1POLA1
SCHEMBL7037704 0.80 NQO2 (0.37) NQO2MTNR1AMTNR1BALDH1A1KDM4E
SCHEMBL7038986 0.77 ABCB1 (0.39) NQO2MTNR1AMTNR1BHTR2AHTR2C
SCHEMBL7037226 0.75 PPARD (0.47) HTR2CPPARD
SCHEMBL7037093 0.75 MTNR1A (0.50) NQO2MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0888309-B1 IMIDAZOLE DERIVATIVES HAVING AFFINITY FOR ALPHA2 RECEPTORS ACTIVITY ORION CORP (FI) 2003-03-19 EP disclosed
US-6313311-B1 ADRENERGIC STIMULANTS FOR POTENTIATING ANESTHETICS PRIOR TO SURGERY; HYPOTENSIVE AGENTS, ANALGESICS, ANTIISCHEMIC AGENTS; NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS ORION CORPORATION (FI) 2001-11-06 US disclosed
EP-0888309-A1 IMIDAZOLE DERIVATIVES HAVING AFFINITY FOR ALPHA2 RECEPTORS ACTIVITY ORION CORPORATION (FI) 1999-01-07 EP disclosed
WO-1997012874-A1 IMIDAZOLE DERIVATIVES HAVING AFFINITY FOR ALPHA2 RECEPTORS ACTIVITY Orion-Yhtymä Oy (FI) 1997-04-10 WO disclosed