SCHEMBL7040941

SCHEMBL7040941

CCCN1CCC(c2nc3c(OC(N)=O)cccc3n2CCN)CC1

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 7/20 0.57
PARP2 Q9UGN5 1/20 0.45
JAK2 O60674 2/20 0.42
JAK1 P23458 2/20 0.42
TYK2 P29597 2/20 0.42
JAK3 P52333 2/20 0.42
HRH1 P35367 8/20 0.42
DRD2 P14416 2/20 0.40
BRD4 O60885 1/20 0.39
CREBBP Q92793 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7035297 0.95 PARP1 (0.52) PARP1PARP2JAK2JAK1TYK2
SCHEMBL7043682 0.92 PARP1 (0.57) PARP1PARP2JAK2JAK1TYK2
SCHEMBL7043338 0.92 PARP1 (0.59) PARP1PARP2HRH1DRD2BRD4
SCHEMBL7046731 0.91 PARP1 (0.56) PARP1PARP2HRH1DRD2BRD4
SCHEMBL7042194 0.91 PARP1 (0.47) PARP1JAK2JAK1TYK2JAK3
SCHEMBL7042083 0.90 PARP1 (0.56) PARP1PARP2HRH1DRD2BRD4
SCHEMBL7042613 0.90 PARP1 (0.56) PARP1PARP2HRH1DRD2BRD4
SCHEMBL7041972 0.90 PARP1 (0.55) PARP1PARP2HRH1DRD2BRD4
SCHEMBL7043782 0.88 PARP1 (0.52) PARP1PARP2HRH1DRD2BRD4
SCHEMBL7042319 0.87 PARP1 (0.52) PARP1PARP2JAK2JAK1TYK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed