SCHEMBL7042340

SCHEMBL7042340

[CH2]C(=O)N(OCC=C)[C@H](C)C(=O)OCc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.42
HCAR2 Q8TDS4 1/20 0.41
LMNA P02545 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
CTSB P07858 2/20 0.39
FAAH O00519 1/20 0.38
MAPK1 P28482 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A3 Q01959 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
CA12 O43570 1/20 0.37
AKR1B10 O60218 1/20 0.37
AKR1B1 P15121 1/20 0.37
CA4 P22748 1/20 0.37
CA6 P23280 1/20 0.37
CA5A P35218 1/20 0.37
CA7 P43166 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5898737 0.89 ALDH1A1 (0.41) ALDH1A1HCAR2LMNAL3MBTL1CTSB
SCHEMBL5898733 0.86 ALDH1A1 (0.39) ALDH1A1HCAR2LMNAL3MBTL1CTSB
Bromide SCHEMBL6315698 0.83 ALDH1A1 (0.36) ALDH1A1HCAR2LMNAL3MBTL1CTSB
SCHEMBL31153792 0.73 ALDH1A1 (0.46) ALDH1A1HCAR2LMNAL3MBTL1CTSB
SCHEMBL26290931 0.73 ALDH1A1 (0.56) ALDH1A1HCAR2LMNAL3MBTL1CTSB
SCHEMBL18510056 0.73 ALDH1A1 (0.56) ALDH1A1HCAR2LMNAL3MBTL1CTSB
SCHEMBL7039395 0.72 CTSB (0.46) ALDH1A1HCAR2CTSBMAPTHPGD
SCHEMBL5898728 0.72 CTSB (0.46) ALDH1A1HCAR2CTSBMAPTHPGD
SCHEMBL7039392 0.72 CTSB (0.46) ALDH1A1HCAR2CTSBMAPTHPGD
SCHEMBL8847794 0.72 ALDH1A1 (0.51) ALDH1A1HCAR2LMNAL3MBTL1CTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003011298-A1 ANTIBACTERIAL OXAZINONES AND METHODS FOR THEIR USE AND SYNTHESIS CHIROLOGIX PHARMACEUTICALS INC. (CA) 2003-02-13 WO disclosed