SCHEMBL7043346

SCHEMBL7043346

CCCN1CCC(c2nc3c(OC(N)=O)cccc3n2CCN2CCCCC2CC)CC1

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.50
PARP2 Q9UGN5 1/20 0.40
HRH1 P35367 6/20 0.38
BRD4 O60885 1/20 0.36
CREBBP Q92793 1/20 0.36
THRB P10828 1/20 0.36
TERT O14746 1/20 0.35
DRD2 P14416 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7039722 0.96 PARP1 (0.45) PARP1PARP2HRH1THRBTERT
SCHEMBL7042195 0.93 PARP1 (0.42) PARP1HRH1THRBDRD2
SCHEMBL7041579 0.90 JAK2 (0.40) PARP1BRD4CREBBPTHRBTERT
SCHEMBL7046731 0.90 PARP1 (0.56) PARP1PARP2HRH1BRD4CREBBP
SCHEMBL7042613 0.89 PARP1 (0.56) PARP1PARP2HRH1BRD4CREBBP
SCHEMBL7041326 0.88 PARP1 (0.43) PARP1THRBTERTDRD2SMN1; SMN2
SCHEMBL7041918 0.88 PARP1 (0.40) PARP1PARP2THRBTERTSMN1; SMN2
SCHEMBL5619904 0.87 PARP1 (0.67) PARP1PARP2HRH1THRBTERT
SCHEMBL7043890 0.87 PARP1 (0.35) PARP1HRH1THRBTERTSMN1; SMN2
SCHEMBL7046819 0.86 CHRM1 (0.40) PARP1PARP2HRH1TERTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed