SCHEMBL7039722

SCHEMBL7039722

CCCN1CCC(c2nc3c(OC(N)=O)cccc3n2CCN2CCCCC2CC)C1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.45
PARP2 Q9UGN5 1/20 0.37
THRB P10828 1/20 0.36
DRD2 P14416 1/20 0.36
DRD3 P35462 1/20 0.36
TERT O14746 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
KDM2B Q8NHM5 1/20 0.34
CYP2D6 P10635 3/20 0.34
HRH1 P35367 3/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7042195 0.97 PARP1 (0.42) PARP1THRBDRD2DRD3KDM2B
SCHEMBL7043346 0.96 PARP1 (0.50) PARP1PARP2THRBDRD2TERT
SCHEMBL7043782 0.89 PARP1 (0.52) PARP1PARP2DRD2DRD3KDM2B
SCHEMBL7042142 0.88 PARP1 (0.52) PARP1PARP2DRD2DRD3SMN1; SMN2
SCHEMBL7041326 0.88 PARP1 (0.43) PARP1THRBDRD2TERTSMN1; SMN2
SCHEMBL7041579 0.88 JAK2 (0.40) PARP1THRBTERTSMN1; SMN2CYP2D6
SCHEMBL5622515 0.87 PARP1 (0.61) PARP1PARP2THRBDRD2DRD3
SCHEMBL7043437 0.86 PARP1 (0.49) PARP1PARP2DRD2DRD3KDM2B
SCHEMBL7043890 0.86 PARP1 (0.35) PARP1THRBTERTSMN1; SMN2CYP2D6
SCHEMBL7043532 0.85 PARP1 (0.48) PARP1PARP2DRD2DRD3KDM2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed