SCHEMBL7043396

SCHEMBL7043396

CN(C(=O)c1nc(-c2ccc(Cl)cc2)c(-c2ccc(Cl)cc2)[nH]1)C1CCCCC1

nearest known ligand 0.61

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 6/20 0.61
TSHR P16473 2/20 0.44
HPGD P15428 1/20 0.44
NPC1 O15118 2/20 0.43
MEN1 O00255 1/20 0.43
POLB P06746 1/20 0.43
KMT2A Q03164 1/20 0.43
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41
S1PR1 P21453 1/20 0.41
PYGL P06737 2/20 0.40
ALDH1A1 P00352 2/20 0.40
LMNA P02545 1/20 0.40
HTT P42858 1/20 0.40
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7044199 0.89 S1PR1 (0.52) CNR1TSHRHPGDNPC1MEN1
SCHEMBL7043234 0.88 CNR1 (0.60) CNR1TSHRHPGDNPC1RAB9A
SCHEMBL6552429 0.88 CNR1 (0.63) CNR1NPC1RAB9A
SCHEMBL7044676 0.88 CNR1 (0.54) CNR1TSHRHPGDNPC1MEN1
SCHEMBL7044597 0.88 CNR1 (0.63) CNR1NPC1RAB9A
SCHEMBL7046176 0.88 NPC1 (0.51) CNR1TSHRHPGDNPC1KMT2A
SCHEMBL7044215 0.87 CNR1 (0.61) CNR1NPC1RAB9A
SCHEMBL7044204 0.80 CNR1 (0.58) CNR1TSHRHPGDNPC1PYGL
SCHEMBL7046592 0.79 CNR1 (0.61) CNR1PTGS1PTGS2
SCHEMBL7041060 0.79 CNR1 (0.52) CNR1PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003007887-A2 SUBSTITUTED IMIDAZOLES AS CANNABINOID RECEPTOR MODULATORS MERCK & CO., INC. (US) 2003-01-30 WO claimed
WO-2003007887-A2 SUBSTITUTED IMIDAZOLES AS CANNABINOID RECEPTOR MODULATORS MERCK & CO., INC. (US) 2003-01-30 WO disclosed