SCHEMBL7044872

SCHEMBL7044872

CN(C)CCn1c(C2CCNC2)nc2c(OC(N)=O)cccc21

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 3/20 0.39
JAK1 P23458 3/20 0.39
TYK2 P29597 3/20 0.39
JAK3 P52333 3/20 0.39
CHRM1 P11229 2/20 0.37
HRH1 P35367 2/20 0.37
PARP1 P09874 4/20 0.36
BRD4 O60885 4/20 0.34
CREBBP Q92793 4/20 0.34
POLB P06746 2/20 0.33
CNR2 P34972 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
HIF1A Q16665 1/20 0.33
NPY1R P25929 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7039421 0.95 CHRM1 (0.44) JAK2JAK1TYK2JAK3CHRM1
SCHEMBL7046373 0.94 JAK2 (0.45) JAK2JAK1TYK2JAK3PARP1
SCHEMBL7041387 0.89 JAK2 (0.42) JAK2JAK1TYK2JAK3CHRM1
SCHEMBL7044226 0.89 JAK2 (0.51) JAK2JAK1TYK2JAK3CHRM1
SCHEMBL7044268 0.88 HRH1 (0.41) JAK2JAK1TYK2JAK3CHRM1
SCHEMBL7043328 0.88 JAK2 (0.40) JAK2JAK1TYK2JAK3CHRM1
SCHEMBL5621364 0.86 PARP1 (0.50) JAK2JAK1TYK2JAK3CHRM1
SCHEMBL7042457 0.85 JAK2 (0.39) JAK2JAK1TYK2JAK3CHRM1
SCHEMBL7042033 0.84 NPY1R (0.40) JAK2JAK1TYK2JAK3CHRM1
SCHEMBL7043077 0.84 PARP1 (0.44) JAK2JAK1TYK2JAK3CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed