SCHEMBL7043328

SCHEMBL7043328

CCn1c(C2CCNC2)nc2c(OC(N)=O)cccc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 3/20 0.40
JAK1 P23458 3/20 0.40
TYK2 P29597 3/20 0.40
JAK3 P52333 3/20 0.40
PARP1 P09874 9/20 0.39
CHRM1 P11229 3/20 0.37
HRH1 P35367 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.34
PARP2 Q9UGN5 3/20 0.33
PARP3 Q9Y6F1 3/20 0.33
ACSS2 Q9NR19 1/20 0.33
MAPK14 Q16539 1/20 0.33
IRAK4 Q9NWZ3 1/20 0.33
TNKS O95271 1/20 0.33
CHRM2 P08172 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
ADRA1A P35348 1/20 0.33
SLC6A3 Q01959 1/20 0.33
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7044486 0.94 CHRM1 (0.44) PARP1CHRM1HRH1PARP2PARP3
SCHEMBL7041855 0.94 JAK2 (0.46) JAK2JAK1TYK2JAK3PARP1
SCHEMBL7044226 0.89 JAK2 (0.51) JAK2JAK1TYK2JAK3PARP1
SCHEMBL7041387 0.89 JAK2 (0.42) JAK2JAK1TYK2JAK3PARP1
SCHEMBL7044268 0.88 HRH1 (0.41) JAK2JAK1TYK2JAK3PARP1
SCHEMBL7044872 0.88 JAK2 (0.39) JAK2JAK1TYK2JAK3PARP1
SCHEMBL7043077 0.86 PARP1 (0.44) JAK2JAK1TYK2JAK3PARP1
SCHEMBL7042457 0.85 JAK2 (0.39) JAK2JAK1TYK2JAK3PARP1
SCHEMBL7042033 0.85 NPY1R (0.40) JAK2JAK1TYK2JAK3PARP1
SCHEMBL5621424 0.84 PARP1 (0.54) JAK2JAK1TYK2JAK3PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed