SCHEMBL7045425

SCHEMBL7045425

[CH2]c1ccc(-c2cnccc2-c2cccc(Cl)c2)cc1F

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
RPS6KA3 P51812 13/20 0.49
LIMK1 P53667 1/20 0.43
NUDT1 P36639 2/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
GCGR P47871 1/20 0.41
MAPK14 Q16539 1/20 0.41
CYP17A1 P05093 1/20 0.40
KDR P35968 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7045431 0.84 RPS6KA3 (0.55) RPS6KA3LIMK1NUDT1KDM4EALDH1A1
SCHEMBL6729132 0.78 RPS6KA3 (0.44) RPS6KA3LIMK1NUDT1KDM4EALDH1A1
SCHEMBL6736780 0.77 RPS6KA3 (0.51) RPS6KA3LIMK1NUDT1KDM4EALDH1A1
SCHEMBL6744643 0.73 RPS6KA3 (0.56) RPS6KA3CYP17A1
SCHEMBL6735505 0.70 NR1H2 (0.43) RPS6KA3LIMK1NUDT1KDM4EALDH1A1
SCHEMBL6646252 0.68 CYP19A1 (0.55) RPS6KA3KDM4ESMN1; SMN2GCGRMAPK14
SCHEMBL6744647 0.68 RPS6KA3 (0.63) RPS6KA3CYP17A1
SCHEMBL7111626 0.68 RPS6KA3 (0.46) RPS6KA3
SCHEMBL7396406 0.67 SLC22A12 (0.54) RPS6KA3LIMK1MAPK14CYP17A1KDR
SCHEMBL6729704 0.67 RPS6KA3 (0.44) RPS6KA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1296971-A2 2-FLUOROBENZENESULFONYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION Pharmacia Corporation (US) 2003-04-02 EP disclosed
WO-2001081332-A2 2-FLUOROBENZENESULFONYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION PHARMACIA CORPORATION (US) 2001-11-01 WO disclosed