SCHEMBL7047642

SCHEMBL7047642

COc1cc(/C=C/c2ccncc2)cc(OC)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 8/20 1.00
CYP1B1 Q16678 8/20 1.00
CYP1A2 P05177 5/20 1.00
KDM4E B2RXH2 2/20 0.71
NPC1 O15118 2/20 0.71
RAB9A P51151 2/20 0.71
CYP2D6 P10635 2/20 0.71
HPGD P15428 2/20 0.71
SMN1; SMN2 Q16637 2/20 0.71
CYP3A4 P08684 1/20 0.71
CYP2C9 P11712 1/20 0.71
CYP2C19 P33261 1/20 0.71
ROCK2 O75116 1/20 0.71
MAP4K4 O95819 1/20 0.71
PRKACA P17612 1/20 0.71
ROCK1 Q13464 1/20 0.71
DYRK1A Q13627 1/20 0.71
NTRK3 Q16288 1/20 0.71
PKN2 Q16513 1/20 0.71
CLK4 Q9HAZ1 1/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7047647 1.00 CYP1A1 (1.00) CYP1A1CYP1B1CYP1A2KDM4ENPC1
SCHEMBL9605438 0.89 CYP1A1 (0.80) CYP1A1CYP1B1CYP1A2KDM4ENPC1
SCHEMBL22594971 0.84 CYP1A1 (0.71) CYP1A1CYP1B1CYP1A2KDM4ENPC1
SCHEMBL8050491 0.83 CYP1A2 (1.00) CYP1A1CYP1B1CYP1A2KDM4ENPC1
SCHEMBL8046590 0.83 CYP1A2 (1.00) CYP1A1CYP1B1CYP1A2KDM4ENPC1
SCHEMBL6833668 0.83 ROCK2 (1.00) CYP1A1CYP1B1CYP1A2KDM4ENPC1
SCHEMBL1743365 0.82 CYP1A1 (1.00) CYP1A1CYP1B1CYP1A2KDM4ENPC1
SCHEMBL1743363 0.82 CYP1A1 (1.00) CYP1A1CYP1B1CYP1A2KDM4ENPC1
SCHEMBL22009168 0.82 CYP1A1 (0.69) CYP1A1CYP1B1CYP1A2KDM4ENPC1
Trismethoxyresveratrol SCHEMBL918739 0.81 CYP1A1 (1.00) CYP1A1CYP1B1CYP1A2KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118530166-A Azastilbene compounds and application thereof in prevention and treatment of metabolic syndrome 中国医学科学院药物研究所 2024-08-23 CN claimed
CN-118530166-A Azastilbene compounds and application thereof in prevention and treatment of metabolic syndrome 中国医学科学院药物研究所 2024-08-23 CN disclosed
WO-2003018013-A1 STILBENE DERIVATIVE HAVING CYTOCHROME P450 1B1 INHIBITORY ACTIVITY, PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, METHOD FOR PREPARING THE SAME, AND COMPOSITION INCLUDING THE SAME PROMEDITECH, INC. (KR) 2003-03-06 WO disclosed