SCHEMBL7048893

SCHEMBL7048893

CNc1nc(C(=O)NCc2ccc(F)cc2)c(O)c(=O)n1C

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNE1 P15382 1/20 0.55
CCR1 P32246 1/20 0.55
KCNQ1 P51787 1/20 0.55
SMN1; SMN2 Q16637 2/20 0.54
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
LIPG Q9Y5X9 1/20 0.52
KCNH2 Q12809 1/20 0.48
CYP2C9 P11712 1/20 0.48
ERCC1 P07992 1/20 0.47
FEN1 P39748 1/20 0.47
ERCC4 Q92889 1/20 0.47
L3MBTL1 Q9Y468 2/20 0.45
TP53 P04637 2/20 0.45
LMNA P02545 1/20 0.45
POLB P06746 1/20 0.45
EGLN1 Q9GZT9 1/20 0.44
SCD O00767 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27635508 0.84 KCNE1 (0.55) KCNE1CCR1KCNQ1SMN1; SMN2MEN1
SCHEMBL6094780 0.83 LIPG (0.42) KCNE1CCR1KCNQ1SMN1; SMN2MEN1
SCHEMBL5314622 0.83 KCNE1 (0.67) KCNE1CCR1KCNQ1SMN1; SMN2MEN1
SCHEMBL13041229 0.82 KCNE1 (0.69) KCNE1CCR1KCNQ1SMN1; SMN2MEN1
SCHEMBL6094550 0.82 KCNH2 (0.54) KCNE1CCR1KCNQ1SMN1; SMN2MEN1
SCHEMBL6094737 0.82 CYP2C9 (0.56) KCNE1CCR1KCNQ1SMN1; SMN2MEN1
SCHEMBL6017760 0.82 SMN1; SMN2 (0.57) KCNE1CCR1KCNQ1SMN1; SMN2MEN1
SCHEMBL1150575 0.82 KCNE1 (0.56) KCNE1CCR1KCNQ1SMN1; SMN2MEN1
SCHEMBL1150195 0.82 KCNE1 (0.56) KCNE1CCR1KCNQ1SMN1; SMN2MEN1
SCHEMBL12776746 0.81 CYP2C9 (0.55) KCNE1CCR1KCNQ1SMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004062613-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-07-29 WO disclosed