SCHEMBL7049865

SCHEMBL7049865

Cc1c(-c2ccccc2)oc2c(C(=O)NCCCN3CCN(c4ccccc4OS(=O)(=O)C(F)(F)F)CC3)cccc2c1=O

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.80
ADRA1A P35348 6/20 0.80
ADRA1D P25100 5/20 0.80
ADRA1B P35368 5/20 0.80
LMNA P02545 2/20 0.54
ALDH1A1 P00352 1/20 0.54
DRD3 P35462 5/20 0.50
SLC6A2 P23975 2/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
KDM4E B2RXH2 1/20 0.50
CYP1A2 P05177 1/20 0.50
CHRM2 P08172 1/20 0.50
CYP3A4 P08684 1/20 0.50
ADRA2A P08913 1/20 0.50
ADORA3 P0DMS8 1/20 0.50
CYP2D6 P10635 1/20 0.50
CHRM1 P11229 1/20 0.50
ACHE P22303 1/20 0.50
PDE4A P27815 1/20 0.50
OPRM1 P35372 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7053164 0.99 HTR1A (0.79) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL7052255 0.92 HTR1A (0.68) HTR1AADRA1AADRA1DADRA1BLMNA
Hydrochloric Acid SCHEMBL7054302 0.91 HTR1A (0.67) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL7047569 0.91 HTR1A (0.83) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL7678716 0.89 HTR1A (0.81) HTR1AADRA1AADRA1DADRA1BLMNA
Upidosin SCHEMBL8907074 0.89 HTR1A (0.94) HTR1AADRA1AADRA1DADRA1BLMNA
Upidosin SCHEMBL29387625 0.89 HTR1A (1.00) HTR1AADRA1AADRA1DADRA1BLMNA
Upidosin SCHEMBL6638869 0.89 HTR1A (1.00) HTR1AADRA1AADRA1DADRA1BLMNA
Upidosin SCHEMBL8908584 0.89 HTR1A (0.93) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL8875547 0.88 HTR1A (0.91) HTR1AADRA1AADRA1DADRA1BLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1222183-B1 BENZOPYRAN DERIVATIVES RECORDATI CHEM PHARM (IT) 2003-04-23 EP claimed
EP-1222183-A1 BENZOPYRAN DERIVATIVES RECORDATI INDUSTRIA CHIMICA E FARMACEUTICA S.p.a. (IT) 2002-07-17 EP claimed
US-6403594-B1 UROGENTIAL INFECTIONS, ETC RECORDATI, S.A. CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 2002-06-11 US claimed
WO-2001029022-A1 BENZOPYRAN DERIVATIVES RECORDATI INDUSTRIA CHIMICA E FARMACEUTICA SPA (IT) 2001-04-26 WO claimed