SCHEMBL7052255

SCHEMBL7052255

Cc1c(-c2ccccc2)oc2c(C(=O)NCCCN3CCN(c4cc(Cl)ccc4OS(=O)(=O)C(F)(F)F)CC3)cccc2c1=O

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.68
ADRA1A P35348 6/20 0.68
ADRA1D P25100 5/20 0.68
ADRA1B P35368 5/20 0.68
LMNA P02545 3/20 0.53
ALDH1A1 P00352 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
MAPT P10636 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
HTR2A P28223 3/20 0.47
HTR2C P28335 3/20 0.47
SLC6A4 P31645 3/20 0.47
KDM4E B2RXH2 2/20 0.47
CYP1A2 P05177 1/20 0.47
CHRM2 P08172 1/20 0.47
CYP3A4 P08684 1/20 0.47
ADRA2A P08913 1/20 0.47
ADORA3 P0DMS8 1/20 0.47
CYP2D6 P10635 1/20 0.47
CHRM1 P11229 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7054302 0.99 HTR1A (0.67) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL7049865 0.92 HTR1A (0.80) HTR1AADRA1AADRA1DADRA1BLMNA
Hydrochloric Acid SCHEMBL7053164 0.91 HTR1A (0.79) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL7054044 0.90 HTR1A (0.69) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL8875520 0.90 HTR1A (0.84) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL7048055 0.90 HTR1A (0.53) HTR1AADRA1AADRA1DADRA1BSMN1; SMN2
SCHEMBL8876429 0.88 HTR1A (0.71) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL8875767 0.86 HTR1A (0.77) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL7051606 0.86 HTR1A (0.72) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL7048075 0.84 HTR1A (0.80) HTR1AADRA1AADRA1DADRA1BLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1222183-B1 BENZOPYRAN DERIVATIVES RECORDATI CHEM PHARM (IT) 2003-04-23 EP claimed
EP-1222183-A1 BENZOPYRAN DERIVATIVES RECORDATI INDUSTRIA CHIMICA E FARMACEUTICA S.p.a. (IT) 2002-07-17 EP claimed
US-6403594-B1 UROGENTIAL INFECTIONS, ETC RECORDATI, S.A. CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 2002-06-11 US claimed
WO-2001029022-A1 BENZOPYRAN DERIVATIVES RECORDATI INDUSTRIA CHIMICA E FARMACEUTICA SPA (IT) 2001-04-26 WO claimed