SCHEMBL7050252

SCHEMBL7050252

CC(C)(C)OC(=O)N1CCC[C@H]1C(=O)NCc1ccc(C#N)cc1Cl

nearest known ligand 0.79

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.79
P2RX7 Q99572 5/20 0.56
LMNA P02545 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
F2 P00734 6/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
NPC1 O15118 1/20 0.48
F10 P00742 2/20 0.47
PRSS1 P07477 2/20 0.47
PRSS2 P07478 2/20 0.47
PRSS3 P35030 2/20 0.47
POLB P06746 1/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
F12 P00748 1/20 0.45
F7 P08709 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7047070 0.88 ALDH1A1 (0.64) ALDH1A1P2RX7LMNANPSR1F2
SCHEMBL7049069 0.85 ALDH1A1 (0.59) ALDH1A1LMNANPSR1F2SMN1; SMN2
SCHEMBL30924055 0.83 EPHX2 (0.58) ALDH1A1P2RX7
SCHEMBL5901213 0.83 ALDH1A1 (0.55) ALDH1A1LMNANPSR1SMN1; SMN2NPC1
SCHEMBL3931937 0.82 ALDH1A1 (0.56) ALDH1A1LMNANPSR1F2SMN1; SMN2
SCHEMBL21520159 0.80 ALDH1A1 (0.52) ALDH1A1LMNANPSR1SMN1; SMN2NPC1
SCHEMBL21520161 0.80 ALDH1A1 (0.52) ALDH1A1LMNANPSR1SMN1; SMN2NPC1
SCHEMBL13111226 0.79 ALDH1A1 (0.51) ALDH1A1LMNANPSR1F2SMN1; SMN2
SCHEMBL21545096 0.79 ALDH1A1 (0.69) ALDH1A1P2RX7LMNANPSR1SMN1; SMN2
SCHEMBL18573086 0.79 ALDH1A1 (0.69) ALDH1A1P2RX7LMNANPSR1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0773955-B1 NEW THROMBIN INHIBITORS, THEIR PREPARATION AND USE BASF AG (DE) 2003-04-16 EP disclosed
EP-0773955-A1 NEW THROMBIN INHIBITORS, THEIR PREPARATION AND USE BASF AKTIENGESELLSCHAFT (DE) 1997-05-21 EP disclosed
WO-1995035309-A1 NEW THROMBIN INHIBITORS, THEIR PREPARATION AND USE BASF AKTIENGESELLSCHAFT (DE) 1995-12-28 WO disclosed